COSTA, GIOSUE'
COSTA, GIOSUE'
Dipartimento di Scienze della Salute
(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies.
2015-01-01 D'Ascenzio, M; Chimenti, P; Gidaro, Mc; De Monte, C; De Vita, D; Granese, A; Scipione, L; Di Santo, R; Costa, G; Alcaro, S; Yáñez, M; Carradori, S
3-Acetyl-25-diaryl-23-dihydro-134-oxadiazoles: a new scaffold for the selective inhibition of monoamine oxidase B
2011-01-01 Maccioni, E; Alcaro, S; Cirilli, R; Vigo, S; Cardia, Mc; Sanna, Ml; Meleddu, R; Yanez, M; Costa, G; Casu, L; Matyus, P; Distinto, S
A Candidate multi-targeting approach to block the CD98hc oncoprotein
2019-01-01 Lanzillotta, D; Iaccino, E; Artese, A; Mimmi, S; Romeo, I; Dattilo, V; Dagostino, S; Costa, G; Gaudio, E; Alcaro, S; Trapasso, F.
A Comparative Docking Strategy to Identify Polyphenolic Derivatives as Promising Antineoplastic Binders of G-quadruplex DNA c-myc and bcl-2 Sequences
2016-01-01 Costa, G; Rocca, R; Moraca, F; Talarico, C; Romeo, I; Ortuso, F; Artese, A; Alcaro, S
A computer-assisted discovery of novel potential anti-obesity compounds as selective carbonic anhydrase VA inhibitors
2019-01-01 Costa, G.; Carta, F.; Ambrosio, F. A.; Artese, A.; Ortuso, F.; Moraca, F.; Rocca, R.; Romeo, I.; Lupia, A.; Maruca, A.; Bagetta, D.; Catalano, R.; Vullo, D.; Alcaro, S.; Supuran, C. T.
A drug repurposing screening reveals a novel epigenetic activity of hydroxychloroquine.
2019-01-01 Catalano, R; Rocca, Roberta; Juli, Giada; Costa, Giosuè; Maruca, A; Artese, A; Caracciolo, D; Tagliaferri, P; Alcaro, S; Tassone, P; Amodio, N.
A first-in-class Wiskott-Aldrich syndrome protein activator with antitumor activity in hematologic cancers
2024-01-01 Spriano, F.; Sartori, G.; Sgrignani, J.; Barnabei, L.; Arribas, A. J.; Guala, M.; Del Amor, A. M. C.; Tomasso, M. R.; Tarantelli, C.; Cascione, L.; Golino, G.; Riveiro, M. E.; Bortolozzi, R.; Lupia, A.; Paduano, F.; Huguet, S.; Rezai, K.; Rinaldi, A.; Margheriti, F.; Ventura, P.; Guarda, G.; Costa, G.; Rocca, R.; Furlan, A.; Verdonk, L. M.; Innocenti, P.; Martin, N. I.; Viola, G.; Driessen, C.; Zucca, E.; Stathis, A.; Gahtory, D.; Van den Nieuwboer, M.; Bornhauser, B.; Alcaro, S.; Trapasso, F.; Cristobal, S.; Padrick, S. B.; Pazzi, N.; Cavalli, F.; Cavalli, A.; Gaudio, E.; Bertoni, F.
ABCC Transporters Mediate the Vacuolar Accumulation of Crocins in Saffron Stigmas
2019-01-01 Demurtas, O. C.; de Brito Francisco, R.; Diretto, G.; Ferrante, P.; Frusciante, S.; Pietrella, M.; Aprea, G.; Borghi, L.; Feeney, M.; Frigerio, L.; Coricello, A.; Costa, G.; Alcaro, S.; Martinoia, E.; Giuliano, G.
Abstract B122: The CD98hc oncoprotein as a target of new anticancer therapy
2019-01-01 Lanzillotta, Delia; Iaccino, Enrico; Artese, Anna; Mimmi, Selena; D'Agostino, Sabrina; Romeo, Isabella; Cantafio, Patrizia; Dattilo, Vincenzo; Costa, Giosuè; Brescia, Carolina; Gaudio, Eugenio; Alcaro, Stefano; Trapasso, Francesco
Active Components of Essential Oils as Anti-Obesity Potential Drugs Investigated by in Silico Techniques
2016-01-01 Costa, G; Gidaro, Mc; Vullo, D; Supuran, Ct; Alcaro, S
An overview on olfaction in the biological, analytical, computational, and machine learning fields
2024-01-01 Chiera, F.; Costa, G.; Alcaro, S.; Artese, A.
Anti-Multiple Myeloma Potential of Secondary Metabolites from Hibiscus sabdariffa-Part 2
2021-01-01 Malacrida, Alessio; Cavalloro, Valeria; Martino, Emanuela; Costa, Giosuè; Ambrosio, Francesca Alessandra; Alcaro, Stefano; Rigolio, Roberta; Cassetti, Arianna; Miloso, Mariarosaria; Collina, Simona
Application of standard and enhanced sampling approaches on non-canonical structures of DNA and RNA
2017-01-01 Moraca, Federica; Rocca, Roberta; Palazzesi, Ferruccio; Costa, Giosue'; Talarico, Carmine; Limongelli, Vittorio; Parrinello, Michele; Alcaro, Stefano
Aryl ethynyl anthraquinones: a useful platform for targeting telomeric G-quadruplex structures
2014-01-01 Percivalle, C; Sissi, C; Greco, Ml; Musetti, C; Mariani, A; Costa, G; Perrore, Ml; Alcaro, S; Freccero, M.; Artese, A
Back Cover: Hit Identification of a Novel Dual Binder for h-telo/c-myc G-Quadruplex by a Combination of Pharmacophore Structure-Based Virtual Screening and Docking Refinement (ChemMedChem 16/2016)
2016-01-01 Rocca, R; Costa, G; Artese, A; Parrotta, L; Ortuso, F; Maccioni, E; Pinato, O; Greco, Ml; Sissi, C; Alcaro, S; Distinto, S; Moraca, F.
Bioactive compounds of Crocus sativus L. and their semi-synthetic derivatives as promising anti-Helicobacter pylori, anti-malarial and anti-leishmanial agents
2015-01-01 De Monte, C; Bizzarri, B; Gidaro, Mc; Carradori, S; Mollica, A; Luisi, G; Granese, A; Alcaro, S; Costa, G; Basilico, N; Parapini, S; Scaltrito, Mm; Masia, C; Sisto, F
BOPC1 Enantiomers Preparation and HuR Interaction Study. From Molecular Modeling to a Curious DEEP-STD NMR Application
2020-01-01 Volpe, S. D.; Listro, R.; Parafioriti, M.; Di Giacomo, M.; Rossi, D.; Ambrosio, F. A.; Costa, G.; Alcaro, S.; Ortuso, F.; Hirsch, A. K. H.; Vasile, F.; Collina, S.
C-6α- vs C-7α-Substituted Steroidal Aromatase Inhibitors: Which Is Better? Synthesis, Biochemical Evaluation, Docking Studies, and Structure-Activity Relationships.
2019-01-01 Roleira, Fmf; Varela, C; Amaral, C; Costa, Sc; Correia-da-Silva, G; Moraca, F; Costa, G; Alcaro, S; Teixeira, Naa; Tavares da Silva, Ej.
Chemoinformatic database building and in silico hit-identification of potential multi-targeting bioactive compounds extracted from mushroom species
2017-01-01 Maruca, A; Moraca, F; Rocca, R; Molisani, F; Alcaro, F; Gidaro, Mc; Alcaro, S; Costa, G; Ortuso, F
Chromene Derivatives as Selective TERRA G-Quadruplex RNA Binders with Antiproliferative Properties
2022-01-01 Rocca, Roberta; Scionti, Francesca; Nadai, Matteo; Moraca, Federica; Maruca, Annalisa; Costa, Giosuè; Catalano, Raffaella; Juli, Giada; Martino, Maria Teresa Di; Ortuso, Francesco; Alcaro, Stefano; Tagliaferri, Pierosandro; Tassone, Pierfrancesco; Richter, Sara N.; Artese, Anna
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| (Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies. | 1-gen-2015 | D'Ascenzio, M; Chimenti, P; Gidaro, Mc; De Monte, C; De Vita, D; Granese, A; Scipione, L; Di Santo, R; Costa, G; Alcaro, S; Yáñez, M; Carradori, S | |
| 3-Acetyl-25-diaryl-23-dihydro-134-oxadiazoles: a new scaffold for the selective inhibition of monoamine oxidase B | 1-gen-2011 | Maccioni, E; Alcaro, S; Cirilli, R; Vigo, S; Cardia, Mc; Sanna, Ml; Meleddu, R; Yanez, M; Costa, G; Casu, L; Matyus, P; Distinto, S | |
| A Candidate multi-targeting approach to block the CD98hc oncoprotein | 1-gen-2019 | Lanzillotta, D; Iaccino, E; Artese, A; Mimmi, S; Romeo, I; Dattilo, V; Dagostino, S; Costa, G; Gaudio, E; Alcaro, S; Trapasso, F. | |
| A Comparative Docking Strategy to Identify Polyphenolic Derivatives as Promising Antineoplastic Binders of G-quadruplex DNA c-myc and bcl-2 Sequences | 1-gen-2016 | Costa, G; Rocca, R; Moraca, F; Talarico, C; Romeo, I; Ortuso, F; Artese, A; Alcaro, S | |
| A computer-assisted discovery of novel potential anti-obesity compounds as selective carbonic anhydrase VA inhibitors | 1-gen-2019 | Costa, G.; Carta, F.; Ambrosio, F. A.; Artese, A.; Ortuso, F.; Moraca, F.; Rocca, R.; Romeo, I.; Lupia, A.; Maruca, A.; Bagetta, D.; Catalano, R.; Vullo, D.; Alcaro, S.; Supuran, C. T. | |
| A drug repurposing screening reveals a novel epigenetic activity of hydroxychloroquine. | 1-gen-2019 | Catalano, R; Rocca, Roberta; Juli, Giada; Costa, Giosuè; Maruca, A; Artese, A; Caracciolo, D; Tagliaferri, P; Alcaro, S; Tassone, P; Amodio, N. | |
| A first-in-class Wiskott-Aldrich syndrome protein activator with antitumor activity in hematologic cancers | 1-gen-2024 | Spriano, F.; Sartori, G.; Sgrignani, J.; Barnabei, L.; Arribas, A. J.; Guala, M.; Del Amor, A. M. C.; Tomasso, M. R.; Tarantelli, C.; Cascione, L.; Golino, G.; Riveiro, M. E.; Bortolozzi, R.; Lupia, A.; Paduano, F.; Huguet, S.; Rezai, K.; Rinaldi, A.; Margheriti, F.; Ventura, P.; Guarda, G.; Costa, G.; Rocca, R.; Furlan, A.; Verdonk, L. M.; Innocenti, P.; Martin, N. I.; Viola, G.; Driessen, C.; Zucca, E.; Stathis, A.; Gahtory, D.; Van den Nieuwboer, M.; Bornhauser, B.; Alcaro, S.; Trapasso, F.; Cristobal, S.; Padrick, S. B.; Pazzi, N.; Cavalli, F.; Cavalli, A.; Gaudio, E.; Bertoni, F. | |
| ABCC Transporters Mediate the Vacuolar Accumulation of Crocins in Saffron Stigmas | 1-gen-2019 | Demurtas, O. C.; de Brito Francisco, R.; Diretto, G.; Ferrante, P.; Frusciante, S.; Pietrella, M.; Aprea, G.; Borghi, L.; Feeney, M.; Frigerio, L.; Coricello, A.; Costa, G.; Alcaro, S.; Martinoia, E.; Giuliano, G. | |
| Abstract B122: The CD98hc oncoprotein as a target of new anticancer therapy | 1-gen-2019 | Lanzillotta, Delia; Iaccino, Enrico; Artese, Anna; Mimmi, Selena; D'Agostino, Sabrina; Romeo, Isabella; Cantafio, Patrizia; Dattilo, Vincenzo; Costa, Giosuè; Brescia, Carolina; Gaudio, Eugenio; Alcaro, Stefano; Trapasso, Francesco | |
| Active Components of Essential Oils as Anti-Obesity Potential Drugs Investigated by in Silico Techniques | 1-gen-2016 | Costa, G; Gidaro, Mc; Vullo, D; Supuran, Ct; Alcaro, S | |
| An overview on olfaction in the biological, analytical, computational, and machine learning fields | 1-gen-2024 | Chiera, F.; Costa, G.; Alcaro, S.; Artese, A. | |
| Anti-Multiple Myeloma Potential of Secondary Metabolites from Hibiscus sabdariffa-Part 2 | 1-gen-2021 | Malacrida, Alessio; Cavalloro, Valeria; Martino, Emanuela; Costa, Giosuè; Ambrosio, Francesca Alessandra; Alcaro, Stefano; Rigolio, Roberta; Cassetti, Arianna; Miloso, Mariarosaria; Collina, Simona | |
| Application of standard and enhanced sampling approaches on non-canonical structures of DNA and RNA | 1-gen-2017 | Moraca, Federica; Rocca, Roberta; Palazzesi, Ferruccio; Costa, Giosue'; Talarico, Carmine; Limongelli, Vittorio; Parrinello, Michele; Alcaro, Stefano | |
| Aryl ethynyl anthraquinones: a useful platform for targeting telomeric G-quadruplex structures | 1-gen-2014 | Percivalle, C; Sissi, C; Greco, Ml; Musetti, C; Mariani, A; Costa, G; Perrore, Ml; Alcaro, S; Freccero, M.; Artese, A | |
| Back Cover: Hit Identification of a Novel Dual Binder for h-telo/c-myc G-Quadruplex by a Combination of Pharmacophore Structure-Based Virtual Screening and Docking Refinement (ChemMedChem 16/2016) | 1-gen-2016 | Rocca, R; Costa, G; Artese, A; Parrotta, L; Ortuso, F; Maccioni, E; Pinato, O; Greco, Ml; Sissi, C; Alcaro, S; Distinto, S; Moraca, F. | |
| Bioactive compounds of Crocus sativus L. and their semi-synthetic derivatives as promising anti-Helicobacter pylori, anti-malarial and anti-leishmanial agents | 1-gen-2015 | De Monte, C; Bizzarri, B; Gidaro, Mc; Carradori, S; Mollica, A; Luisi, G; Granese, A; Alcaro, S; Costa, G; Basilico, N; Parapini, S; Scaltrito, Mm; Masia, C; Sisto, F | |
| BOPC1 Enantiomers Preparation and HuR Interaction Study. From Molecular Modeling to a Curious DEEP-STD NMR Application | 1-gen-2020 | Volpe, S. D.; Listro, R.; Parafioriti, M.; Di Giacomo, M.; Rossi, D.; Ambrosio, F. A.; Costa, G.; Alcaro, S.; Ortuso, F.; Hirsch, A. K. H.; Vasile, F.; Collina, S. | |
| C-6α- vs C-7α-Substituted Steroidal Aromatase Inhibitors: Which Is Better? Synthesis, Biochemical Evaluation, Docking Studies, and Structure-Activity Relationships. | 1-gen-2019 | Roleira, Fmf; Varela, C; Amaral, C; Costa, Sc; Correia-da-Silva, G; Moraca, F; Costa, G; Alcaro, S; Teixeira, Naa; Tavares da Silva, Ej. | |
| Chemoinformatic database building and in silico hit-identification of potential multi-targeting bioactive compounds extracted from mushroom species | 1-gen-2017 | Maruca, A; Moraca, F; Rocca, R; Molisani, F; Alcaro, F; Gidaro, Mc; Alcaro, S; Costa, G; Ortuso, F | |
| Chromene Derivatives as Selective TERRA G-Quadruplex RNA Binders with Antiproliferative Properties | 1-gen-2022 | Rocca, Roberta; Scionti, Francesca; Nadai, Matteo; Moraca, Federica; Maruca, Annalisa; Costa, Giosuè; Catalano, Raffaella; Juli, Giada; Martino, Maria Teresa Di; Ortuso, Francesco; Alcaro, Stefano; Tagliaferri, Pierosandro; Tassone, Pierfrancesco; Richter, Sara N.; Artese, Anna |