RicercaInizia una nuova ricerca
NOTA: è possibile cercare una corrispondenza esatta usando i doppi apici, ad es: "evoluzione della specie". Qualora si cerchi un identificativo, è consigliabile cercarlo in due modi differenti: tra apici con caratteri speciali es: "978-94-6366-274" oppure senza caratteri speciali solo come sequenza numerica: es 978946366274.
(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro-1H-indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase
2015-01-01 Meleddu, R; Distinto, S; Corona, A; Bianco, G; Cannas, V; Esposito, F; Alcaro, S; Matyus, P; Bogdan, D; Cottiglia, F; Tramontano, E; Maccioni, E; Artese, A
(E)-3-Heteroarylidenechroman-4-ones as potent and selective monoamine oxidase-B inhibitors
2016-01-01 Desideri, N; Proietti Monaco, L; Fioravanti, R; Biava, M; Yáñez, M; Ortuso, F; Alcaro, S
(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies.
2015-01-01 D'Ascenzio, M; Chimenti, P; Gidaro, Mc; De Monte, C; De Vita, D; Granese, A; Scipione, L; Di Santo, R; Costa, G; Alcaro, S; Yáñez, M; Carradori, S
1,5-Diphenylpenta-2,4-dien-1-ones as potent and selective monoamine oxidase-B inhibitors
2013-01-01 Desideri, N; Fioravanti, R; Proietti Monaco, L; Biava, M; Yáñez, M; Ortuso, F; Alcaro, S
1- acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazole; a new scaffold for monoaminoxidase inhibitors: design, synthesis, and biological properties
2008-01-01 Vigo, S; Alcaro, S; Bolasco, A; Cardia, C; Distinto, S; Maccioni, E; Orallo, F; Ortuso, F; Sanna, M. L.; Secci, D; Yanez, M
1-benzenesulfonamide-1(H)-pyrazoles and 3-benzenesulfonamide-4-tiazolidinones, two promising scaffolds for the design of cycloxygenase inhibitors
2008-01-01 SANNA M., L; Alcaro, S; Bolasco, A; Cardia, C; Cirilli, R; Distinto, S; Maccioni, E; Orallo, F; Ortuso, F; Secci, D; Vigo, S; Yanez, M
2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms
2023-01-01 Sequeira, Lisa; Distinto, Simona; Meleddu, Rita; Gaspari, Marco; Angeli, ; Rea, Federico; Cottiglia, Filippo; Secci, Daniela; Onali, Alessia; Sanna, Erica; Borges, Fernanda; Uriarte, Eugenio; Alcaro, Stefano; Supuran, Claudiu T.; Maccioni, Elias
3-Acetyl-25-diaryl-23-dihydro-134-oxadiazoles: a new scaffold for the selective inhibition of monoamine oxidase B
2011-01-01 Maccioni, E; Alcaro, S; Cirilli, R; Vigo, S; Cardia, Mc; Sanna, Ml; Meleddu, R; Yanez, M; Costa, G; Casu, L; Matyus, P; Distinto, S
4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis
2019-01-01 Secci, D; Carradori, S; Petzer, A; Guglielmi, P; D'Ascenzio, M; Chimenti, P; Bagetta, D; Alcaro, S; Zengin, G; Petzer, Jp; Ortuso, F
4-carbossamido-9-fluorenoni: proprietà anti-HSV-2 e immunostimolanti
2004-01-01 Alcaro, S; Arena, A.; DI BELLA, R.; Ortuso, F.; Ottan, R.; Neri, S.; Pavone, B.; Vigorita, M. G.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro-1H-indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase | 1-gen-2015 | Meleddu, R; Distinto, S; Corona, A; Bianco, G; Cannas, V; Esposito, F; Alcaro, S; Matyus, P; Bogdan, D; Cottiglia, F; Tramontano, E; Maccioni, E; Artese, A | |
(E)-3-Heteroarylidenechroman-4-ones as potent and selective monoamine oxidase-B inhibitors | 1-gen-2016 | Desideri, N; Proietti Monaco, L; Fioravanti, R; Biava, M; Yáñez, M; Ortuso, F; Alcaro, S | |
(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies. | 1-gen-2015 | D'Ascenzio, M; Chimenti, P; Gidaro, Mc; De Monte, C; De Vita, D; Granese, A; Scipione, L; Di Santo, R; Costa, G; Alcaro, S; Yáñez, M; Carradori, S | |
1,5-Diphenylpenta-2,4-dien-1-ones as potent and selective monoamine oxidase-B inhibitors | 1-gen-2013 | Desideri, N; Fioravanti, R; Proietti Monaco, L; Biava, M; Yáñez, M; Ortuso, F; Alcaro, S | |
1- acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazole; a new scaffold for monoaminoxidase inhibitors: design, synthesis, and biological properties | 1-gen-2008 | Vigo, S; Alcaro, S; Bolasco, A; Cardia, C; Distinto, S; Maccioni, E; Orallo, F; Ortuso, F; Sanna, M. L.; Secci, D; Yanez, M | |
1-benzenesulfonamide-1(H)-pyrazoles and 3-benzenesulfonamide-4-tiazolidinones, two promising scaffolds for the design of cycloxygenase inhibitors | 1-gen-2008 | SANNA M., L; Alcaro, S; Bolasco, A; Cardia, C; Cirilli, R; Distinto, S; Maccioni, E; Orallo, F; Ortuso, F; Secci, D; Vigo, S; Yanez, M | |
2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms | 1-gen-2023 | Sequeira, Lisa; Distinto, Simona; Meleddu, Rita; Gaspari, Marco; Angeli, ; Rea, Federico; Cottiglia, Filippo; Secci, Daniela; Onali, Alessia; Sanna, Erica; Borges, Fernanda; Uriarte, Eugenio; Alcaro, Stefano; Supuran, Claudiu T.; Maccioni, Elias | |
3-Acetyl-25-diaryl-23-dihydro-134-oxadiazoles: a new scaffold for the selective inhibition of monoamine oxidase B | 1-gen-2011 | Maccioni, E; Alcaro, S; Cirilli, R; Vigo, S; Cardia, Mc; Sanna, Ml; Meleddu, R; Yanez, M; Costa, G; Casu, L; Matyus, P; Distinto, S | |
4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis | 1-gen-2019 | Secci, D; Carradori, S; Petzer, A; Guglielmi, P; D'Ascenzio, M; Chimenti, P; Bagetta, D; Alcaro, S; Zengin, G; Petzer, Jp; Ortuso, F | |
4-carbossamido-9-fluorenoni: proprietà anti-HSV-2 e immunostimolanti | 1-gen-2004 | Alcaro, S; Arena, A.; DI BELLA, R.; Ortuso, F.; Ottan, R.; Neri, S.; Pavone, B.; Vigorita, M. G. |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile
Opzioni
Scopri
Tipologia
- 1 Contributo su Rivista 292
- 1 Contributo su Rivista::1.1 Arti... 284
- 4 Contributo in Atti di Convegno ... 134
- 4 Contributo in Atti di Convegno ... 121
- 5 Altro 42
- 5 Altro::5.12 Altro 42
- 2 Contributo in Volume 9
- 2 Contributo in Volume::2.1 Contr... 9
- 4 Contributo in Atti di Convegno ... 9
- 1 Contributo su Rivista::1.2 Rece... 7
- 4 Contributo in Atti di Convegno ... 4
- 1 Contributo su Rivista::1.5 Abst... 1
- 3 Libro 1
- 3 Libro::3.1 Monografia o trattat... 1
Data di pubblicazione
- In corso di stampa 1
- 2020 - 2023 76
- 2010 - 2019 185
- 2000 - 2009 186
- 1990 - 1999 29
- 1989 - 1989 1
Editore
- Alcaro 1
- Casa Editrice Ambrosiana 1
- COMPUTATIONALLY DRIVEN DRUG DISCO... 1
- Institute of Electrical and Elect... 1
- Missailidis 1
- Research Signpost 1
- UMG 1
- VMD VERLAG 1
- WILEY-BLACKWELL 1
- Wiley-VCH 1
Rivista
- EUROPEAN JOURNAL OF MEDICINAL CHE... 31
- JOURNAL OF MEDICINAL CHEMISTRY 21
- BIOORGANIC & MEDICINAL CHEMISTRY ... 13
- MOLECULES 12
- BIOORGANIC & MEDICINAL CHEMISTRY 11
- EUROPEAN JOURNAL OF MEDICINAL CHE... 10
- JOURNAL OF ENZYME INHIBITION AND ... 9
- CHEMMEDCHEM 7
- ACS MEDICINAL CHEMISTRY LETTERS 6
- ANTIOXIDANTS 6
Serie
- METHODS IN MOLECULAR BIOLOGY 1
Keyword
- Humans 22
- Structure-Activity Relationship 15
- docking 14
- Molecular Structure 14
- Dose-Response Relationship 11
- Drug 11
- Models 10
- Docking 9
- Molecular 9
- Molecular Docking Simulation 7
Lingua
- eng 382
- ita 67
Accesso al fulltext
- no fulltext 478