Sfoglia per Rivista BIOORGANIC
Molecular modeling and enzymatic studies of the interaction of a choline analogue and acetylcholinesterase
2002-01-01 Scipione, L; Ortuso, F; Posca, S; Rispoli, V; Rotiroti, D; Alcaro, S
New 4-[(3-cyclohexyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzene-1-sulfonamides, synthesis and inhibitory activity toward carbonic anhydrase I, II, IX, XII
2015-01-01 Meleddu, R; Maccioni, E; Distinto, S; Bianco, G; Melis, C; Alcaro, S; Cottiglia, F; Ceruso, M; Supuran, Ct
New 7,8-ethylenedioxy-2,3-benzodiazepines as noncompetitive AMPA receptor antagonists
2006-01-01 Zappala, M; Pellicano, A; Micale, N; Menniti, Fs; Ferreri, G; De Sarro, G; Grasso, S; De Micheli, C
New conformationally locked bicyclic N,O-nucleoside analogues of antiviral drugs
2005-01-01 Procopio, A; DE NINO, A; Maiuolo, L; Ortuso, F; Sindona, G; Alcaro, S
Preparation, characterization,molecular modeling and in vitro activity of paclitaxel cyclodextrin complexes
2002-01-01 Ventura, C. A.; Battaglia, D; Ortuso, F; Cattel, L; Puglisi, G; Alcaro, S; Fresta, M; Paolino, D
Quercetin-3-oleoyl derivatives as new GPR40 agonists: Molecular docking studies and functional evaluation
2019-01-01 Carullo, Gabriele; Perri, Mariarita; Manetti, Fabrizio; Aiello, Francesca; Caroleo, Maria Cristina; Cione, Erika
Synthesis and molecular modelling studies of prenylated pyrazolines as MAO-B inhibitors
2010-01-01 Fioravanti, R; Bolasco, A; Manna, F; Rossi, F; Orallo, F; Yáñez, M; Vitali, A; Alcaro, S; Ortuso, F
Synthesis, molecular modeling studies, and selective inhibitory activity against monoamine oxidase of N,N'-bis[2-oxo-2H-benzopyran]-3-carboxamides
2006-01-01 Chimenti, F; Secci, D; Bolasco, A; Chimenti, P; Granese, A; Carradori, S; Befani, O; Turini, P; Ortuso, F; Alcaro, S
Tetraplex DNA specific ligands based on the fluorenone-carboxamide scaffold
2007-01-01 Alcaro, S; Artese, A; Iley, J. N.; Maccari, R; Missailidis, S; Ottana, R; Ragazzon, P; Vigorita, M. G.; Ortuso, F
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Molecular modeling and enzymatic studies of the interaction of a choline analogue and acetylcholinesterase | 1-gen-2002 | Scipione, L; Ortuso, F; Posca, S; Rispoli, V; Rotiroti, D; Alcaro, S | |
New 4-[(3-cyclohexyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzene-1-sulfonamides, synthesis and inhibitory activity toward carbonic anhydrase I, II, IX, XII | 1-gen-2015 | Meleddu, R; Maccioni, E; Distinto, S; Bianco, G; Melis, C; Alcaro, S; Cottiglia, F; Ceruso, M; Supuran, Ct | |
New 7,8-ethylenedioxy-2,3-benzodiazepines as noncompetitive AMPA receptor antagonists | 1-gen-2006 | Zappala, M; Pellicano, A; Micale, N; Menniti, Fs; Ferreri, G; De Sarro, G; Grasso, S; De Micheli, C | |
New conformationally locked bicyclic N,O-nucleoside analogues of antiviral drugs | 1-gen-2005 | Procopio, A; DE NINO, A; Maiuolo, L; Ortuso, F; Sindona, G; Alcaro, S | |
Preparation, characterization,molecular modeling and in vitro activity of paclitaxel cyclodextrin complexes | 1-gen-2002 | Ventura, C. A.; Battaglia, D; Ortuso, F; Cattel, L; Puglisi, G; Alcaro, S; Fresta, M; Paolino, D | |
Quercetin-3-oleoyl derivatives as new GPR40 agonists: Molecular docking studies and functional evaluation | 1-gen-2019 | Carullo, Gabriele; Perri, Mariarita; Manetti, Fabrizio; Aiello, Francesca; Caroleo, Maria Cristina; Cione, Erika | |
Synthesis and molecular modelling studies of prenylated pyrazolines as MAO-B inhibitors | 1-gen-2010 | Fioravanti, R; Bolasco, A; Manna, F; Rossi, F; Orallo, F; Yáñez, M; Vitali, A; Alcaro, S; Ortuso, F | |
Synthesis, molecular modeling studies, and selective inhibitory activity against monoamine oxidase of N,N'-bis[2-oxo-2H-benzopyran]-3-carboxamides | 1-gen-2006 | Chimenti, F; Secci, D; Bolasco, A; Chimenti, P; Granese, A; Carradori, S; Befani, O; Turini, P; Ortuso, F; Alcaro, S | |
Tetraplex DNA specific ligands based on the fluorenone-carboxamide scaffold | 1-gen-2007 | Alcaro, S; Artese, A; Iley, J. N.; Maccari, R; Missailidis, S; Ottana, R; Ragazzon, P; Vigorita, M. G.; Ortuso, F |
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