ALCARO, Stefano
ALCARO, Stefano
Dipartimento di Scienze della Salute
(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro-1H-indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase
2015-01-01 Meleddu, R; Distinto, S; Corona, A; Bianco, G; Cannas, V; Esposito, F; Alcaro, S; Matyus, P; Bogdan, D; Cottiglia, F; Tramontano, E; Maccioni, E; Artese, A
(E)-3-Heteroarylidenechroman-4-ones as potent and selective monoamine oxidase-B inhibitors
2016-01-01 Desideri, N; Proietti Monaco, L; Fioravanti, R; Biava, M; Yáñez, M; Ortuso, F; Alcaro, S
(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies.
2015-01-01 D'Ascenzio, M; Chimenti, P; Gidaro, Mc; De Monte, C; De Vita, D; Granese, A; Scipione, L; Di Santo, R; Costa, G; Alcaro, S; Yáñez, M; Carradori, S
1,5-Diphenylpenta-2,4-dien-1-ones as potent and selective monoamine oxidase-B inhibitors
2013-01-01 Desideri, N; Fioravanti, R; Proietti Monaco, L; Biava, M; Yáñez, M; Ortuso, F; Alcaro, S
1- acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazole; a new scaffold for monoaminoxidase inhibitors: design, synthesis, and biological properties
2008-01-01 Vigo, S; Alcaro, S; Bolasco, A; Cardia, C; Distinto, S; Maccioni, E; Orallo, F; Ortuso, F; Sanna, M. L.; Secci, D; Yanez, M
1-benzenesulfonamide-1(H)-pyrazoles and 3-benzenesulfonamide-4-tiazolidinones, two promising scaffolds for the design of cycloxygenase inhibitors
2008-01-01 SANNA M., L; Alcaro, S; Bolasco, A; Cardia, C; Cirilli, R; Distinto, S; Maccioni, E; Orallo, F; Ortuso, F; Secci, D; Vigo, S; Yanez, M
2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms
2023-01-01 Sequeira, Lisa; Distinto, Simona; Meleddu, Rita; Gaspari, Marco; Angeli, Andrea; Cottiglia, Filippo; Secci, Daniela; Onali, Alessia; Sanna, Erica; Borges, Fernanda; Uriarte, Eugenio; Alcaro, Stefano; Supuran, Claudiu T.; Maccioni, Elias
3-Acetyl-25-diaryl-23-dihydro-134-oxadiazoles: a new scaffold for the selective inhibition of monoamine oxidase B
2011-01-01 Maccioni, E; Alcaro, S; Cirilli, R; Vigo, S; Cardia, Mc; Sanna, Ml; Meleddu, R; Yanez, M; Costa, G; Casu, L; Matyus, P; Distinto, S
4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis
2019-01-01 Secci, D; Carradori, S; Petzer, A; Guglielmi, P; D'Ascenzio, M; Chimenti, P; Bagetta, D; Alcaro, S; Zengin, G; Petzer, Jp; Ortuso, F
4-carbossamido-9-fluorenoni: proprietà anti-HSV-2 e immunostimolanti
2004-01-01 Alcaro, S; Arena, A.; DI BELLA, R.; Ortuso, F.; Ottan, R.; Neri, S.; Pavone, B.; Vigorita, M. G.
4-Oxoquinolines and monoamine oxidase: When tautomerism matters
2021-01-01 Mesiti, Francesco; Maruca, Annalisa; Silva, Vera; Rocca, Roberta; Fernandes, Carlos; Remião, Fernando; Uriarte, Eugenio; Alcaro, Stefano; Gaspar, Alexandra; Borges, Fernanda
8-Amide and 8-carbamate substitution patterns as modulators of 7-hydroxy-4-methylcoumarin's antidepressant profile: Synthesis, biological evaluation and docking studies
2023-01-01 Matos, M. J.; Novo, P.; Mayan, L.; Torres, I.; Uriarte, E.; Yanez, M.; Fontenla, J. A.; Ortuso, F.; Alcaro, S.; Procopio, F.; Rodriguez-Franco, M. I.; Val, C.; Loza, M. I.; Brea, J.; Borges, F.; Vina, D.
8-Amide and 8-Carbamate Substitution Patterns as Modulators of 7-Hydroxy-4-Methylcoumarin{'}s Antidepressant Profile: Synthesis, MAO Inhibition, Cytotoxicity and Docking Studies
2022-01-01 Matos, M. J.; Novo, P.; May('a)n, L.; Torres, I.; Uriarte, E.; Y('a)(\~n)ez, M.; Fontenla, J. ?.; Ortuso, F.; Alcaro, S.; Procopio, F.; Borges, F.; Vi(\~n)a, D.
9-fluorenon-4-carboxamides: synthesis, conformational analysis, anti-HSV-2, and immunomodulatory evaluation. Note II
2004-01-01 Arena, A; DI BELLA, R; Neri, S; Ottanà, R; Ortuso, F; Pavone, B; Vigorita, M. G.; Alcaro, S
A "Quasi-Flexible" Automatic Docking Processing for Studying Stereoselective Recognition Mechanisms. Part I. Protocol Validation
2000-01-01 Alcaro, S.; Gasparrini, F.; Incani, O.; Mecucci, S.; Misiti, D.; Pierini, M.; Villani, C.
A Candidate multi-targeting approach to block the CD98hc oncoprotein
2019-01-01 Lanzillotta, D; Iaccino, E; Artese, A; Mimmi, S; Romeo, I; Dattilo, V; Dagostino, S; Costa, G; Gaudio, E; Alcaro, S; Trapasso, F.
A chromatographic and computational study on the driving force operating in the exceptionally large enantioseparation of N-thiocarbamoyl-3-(4'-biphenyl)-5-phenyl-4,5-dihydro-(1H) pyrazole on a 4-methylbenzoate cellulose-based chiral stationary phase
2014-01-01 Alcaro, S; Menta, S; Fioravanti, R; Cirilli, R; Ortuso, F
A chromatographic study on the exceptional enantioselectivity of cellulose tris(4-methylbenzoate) towards C5-chiral 45-dihydro-(1H)-pyrazole derivatives
2011-01-01 Cirilli, R; Alcaro, S; Fioravanti, R; Ferretti, R; Bolasco, A; Gallinella, B; Faggi, C
A Comparative Docking Strategy to Identify Polyphenolic Derivatives as Promising Antineoplastic Binders of G-quadruplex DNA c-myc and bcl-2 Sequences
2016-01-01 Costa, G; Rocca, R; Moraca, F; Talarico, C; Romeo, I; Ortuso, F; Artese, A; Alcaro, S
A comparative study of the in vitro inhibitory activity of tacrine-like molecules (Paraquat, MPTP, MPDP and MPP+) on hydrolysis by acetylcholine and butyrylcholine esterases
2004-01-01 Arcone, R.; Alcaro, S; Battaglia, D.; Gallelli, A.; Iannone, M.; Rotiroti, D.; Vecchio, I.; Ortuso, F
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro-1H-indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase | 1-gen-2015 | Meleddu, R; Distinto, S; Corona, A; Bianco, G; Cannas, V; Esposito, F; Alcaro, S; Matyus, P; Bogdan, D; Cottiglia, F; Tramontano, E; Maccioni, E; Artese, A | |
(E)-3-Heteroarylidenechroman-4-ones as potent and selective monoamine oxidase-B inhibitors | 1-gen-2016 | Desideri, N; Proietti Monaco, L; Fioravanti, R; Biava, M; Yáñez, M; Ortuso, F; Alcaro, S | |
(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies. | 1-gen-2015 | D'Ascenzio, M; Chimenti, P; Gidaro, Mc; De Monte, C; De Vita, D; Granese, A; Scipione, L; Di Santo, R; Costa, G; Alcaro, S; Yáñez, M; Carradori, S | |
1,5-Diphenylpenta-2,4-dien-1-ones as potent and selective monoamine oxidase-B inhibitors | 1-gen-2013 | Desideri, N; Fioravanti, R; Proietti Monaco, L; Biava, M; Yáñez, M; Ortuso, F; Alcaro, S | |
1- acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazole; a new scaffold for monoaminoxidase inhibitors: design, synthesis, and biological properties | 1-gen-2008 | Vigo, S; Alcaro, S; Bolasco, A; Cardia, C; Distinto, S; Maccioni, E; Orallo, F; Ortuso, F; Sanna, M. L.; Secci, D; Yanez, M | |
1-benzenesulfonamide-1(H)-pyrazoles and 3-benzenesulfonamide-4-tiazolidinones, two promising scaffolds for the design of cycloxygenase inhibitors | 1-gen-2008 | SANNA M., L; Alcaro, S; Bolasco, A; Cardia, C; Cirilli, R; Distinto, S; Maccioni, E; Orallo, F; Ortuso, F; Secci, D; Vigo, S; Yanez, M | |
2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms | 1-gen-2023 | Sequeira, Lisa; Distinto, Simona; Meleddu, Rita; Gaspari, Marco; Angeli, Andrea; Cottiglia, Filippo; Secci, Daniela; Onali, Alessia; Sanna, Erica; Borges, Fernanda; Uriarte, Eugenio; Alcaro, Stefano; Supuran, Claudiu T.; Maccioni, Elias | |
3-Acetyl-25-diaryl-23-dihydro-134-oxadiazoles: a new scaffold for the selective inhibition of monoamine oxidase B | 1-gen-2011 | Maccioni, E; Alcaro, S; Cirilli, R; Vigo, S; Cardia, Mc; Sanna, Ml; Meleddu, R; Yanez, M; Costa, G; Casu, L; Matyus, P; Distinto, S | |
4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis | 1-gen-2019 | Secci, D; Carradori, S; Petzer, A; Guglielmi, P; D'Ascenzio, M; Chimenti, P; Bagetta, D; Alcaro, S; Zengin, G; Petzer, Jp; Ortuso, F | |
4-carbossamido-9-fluorenoni: proprietà anti-HSV-2 e immunostimolanti | 1-gen-2004 | Alcaro, S; Arena, A.; DI BELLA, R.; Ortuso, F.; Ottan, R.; Neri, S.; Pavone, B.; Vigorita, M. G. | |
4-Oxoquinolines and monoamine oxidase: When tautomerism matters | 1-gen-2021 | Mesiti, Francesco; Maruca, Annalisa; Silva, Vera; Rocca, Roberta; Fernandes, Carlos; Remião, Fernando; Uriarte, Eugenio; Alcaro, Stefano; Gaspar, Alexandra; Borges, Fernanda | |
8-Amide and 8-carbamate substitution patterns as modulators of 7-hydroxy-4-methylcoumarin's antidepressant profile: Synthesis, biological evaluation and docking studies | 1-gen-2023 | Matos, M. J.; Novo, P.; Mayan, L.; Torres, I.; Uriarte, E.; Yanez, M.; Fontenla, J. A.; Ortuso, F.; Alcaro, S.; Procopio, F.; Rodriguez-Franco, M. I.; Val, C.; Loza, M. I.; Brea, J.; Borges, F.; Vina, D. | |
8-Amide and 8-Carbamate Substitution Patterns as Modulators of 7-Hydroxy-4-Methylcoumarin{'}s Antidepressant Profile: Synthesis, MAO Inhibition, Cytotoxicity and Docking Studies | 1-gen-2022 | Matos, M. J.; Novo, P.; May('a)n, L.; Torres, I.; Uriarte, E.; Y('a)(\~n)ez, M.; Fontenla, J. ?.; Ortuso, F.; Alcaro, S.; Procopio, F.; Borges, F.; Vi(\~n)a, D. | |
9-fluorenon-4-carboxamides: synthesis, conformational analysis, anti-HSV-2, and immunomodulatory evaluation. Note II | 1-gen-2004 | Arena, A; DI BELLA, R; Neri, S; Ottanà, R; Ortuso, F; Pavone, B; Vigorita, M. G.; Alcaro, S | |
A "Quasi-Flexible" Automatic Docking Processing for Studying Stereoselective Recognition Mechanisms. Part I. Protocol Validation | 1-gen-2000 | Alcaro, S.; Gasparrini, F.; Incani, O.; Mecucci, S.; Misiti, D.; Pierini, M.; Villani, C. | |
A Candidate multi-targeting approach to block the CD98hc oncoprotein | 1-gen-2019 | Lanzillotta, D; Iaccino, E; Artese, A; Mimmi, S; Romeo, I; Dattilo, V; Dagostino, S; Costa, G; Gaudio, E; Alcaro, S; Trapasso, F. | |
A chromatographic and computational study on the driving force operating in the exceptionally large enantioseparation of N-thiocarbamoyl-3-(4'-biphenyl)-5-phenyl-4,5-dihydro-(1H) pyrazole on a 4-methylbenzoate cellulose-based chiral stationary phase | 1-gen-2014 | Alcaro, S; Menta, S; Fioravanti, R; Cirilli, R; Ortuso, F | |
A chromatographic study on the exceptional enantioselectivity of cellulose tris(4-methylbenzoate) towards C5-chiral 45-dihydro-(1H)-pyrazole derivatives | 1-gen-2011 | Cirilli, R; Alcaro, S; Fioravanti, R; Ferretti, R; Bolasco, A; Gallinella, B; Faggi, C | |
A Comparative Docking Strategy to Identify Polyphenolic Derivatives as Promising Antineoplastic Binders of G-quadruplex DNA c-myc and bcl-2 Sequences | 1-gen-2016 | Costa, G; Rocca, R; Moraca, F; Talarico, C; Romeo, I; Ortuso, F; Artese, A; Alcaro, S | |
A comparative study of the in vitro inhibitory activity of tacrine-like molecules (Paraquat, MPTP, MPDP and MPP+) on hydrolysis by acetylcholine and butyrylcholine esterases | 1-gen-2004 | Arcone, R.; Alcaro, S; Battaglia, D.; Gallelli, A.; Iannone, M.; Rotiroti, D.; Vecchio, I.; Ortuso, F |