ORTUSO, Francesco
ORTUSO, Francesco
Dipartimento di Scienze della Salute
"Synthesis, Biological Evaluation and Molecular Modeling of Natural and Semi-synthetic Oleuropeine Drivates as Cox-l and -2 Inhibitors
2008-01-01 Procopio, Antonio; Stefano, Alcaro; Ortuso, Francesco; Nardi, M; Giovanni, Sindona; Paolo, Sacchelta; Oliverio, Manuela
(E)-3-Heteroarylidenechroman-4-ones as potent and selective monoamine oxidase-B inhibitors
2016-01-01 Desideri, N; Proietti Monaco, L; Fioravanti, R; Biava, M; Yáñez, M; Ortuso, F; Alcaro, S
1,5-Diphenylpenta-2,4-dien-1-ones as potent and selective monoamine oxidase-B inhibitors
2013-01-01 Desideri, N; Fioravanti, R; Proietti Monaco, L; Biava, M; Yáñez, M; Ortuso, F; Alcaro, S
1- acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazole; a new scaffold for monoaminoxidase inhibitors: design, synthesis, and biological properties
2008-01-01 Vigo, S; Alcaro, S; Bolasco, A; Cardia, C; Distinto, S; Maccioni, E; Orallo, F; Ortuso, F; Sanna, M. L.; Secci, D; Yanez, M
1-benzenesulfonamide-1(H)-pyrazoles and 3-benzenesulfonamide-4-tiazolidinones, two promising scaffolds for the design of cycloxygenase inhibitors
2008-01-01 SANNA M., L; Alcaro, S; Bolasco, A; Cardia, C; Cirilli, R; Distinto, S; Maccioni, E; Orallo, F; Ortuso, F; Secci, D; Vigo, S; Yanez, M
4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis
2019-01-01 Secci, D; Carradori, S; Petzer, A; Guglielmi, P; D'Ascenzio, M; Chimenti, P; Bagetta, D; Alcaro, S; Zengin, G; Petzer, Jp; Ortuso, F
4-carbossamido-9-fluorenoni: proprietà anti-HSV-2 e immunostimolanti
2004-01-01 Alcaro, S; Arena, A.; DI BELLA, R.; Ortuso, F.; Ottan, R.; Neri, S.; Pavone, B.; Vigorita, M. G.
8-Amide and 8-carbamate substitution patterns as modulators of 7-hydroxy-4-methylcoumarin's antidepressant profile: Synthesis, biological evaluation and docking studies
2023-01-01 Matos, M. J.; Novo, P.; Mayan, L.; Torres, I.; Uriarte, E.; Yanez, M.; Fontenla, J. A.; Ortuso, F.; Alcaro, S.; Procopio, F.; Rodriguez-Franco, M. I.; Val, C.; Loza, M. I.; Brea, J.; Borges, F.; Vina, D.
8-Amide and 8-Carbamate Substitution Patterns as Modulators of 7-Hydroxy-4-Methylcoumarin{'}s Antidepressant Profile: Synthesis, MAO Inhibition, Cytotoxicity and Docking Studies
2022-01-01 Matos, M. J.; Novo, P.; May('a)n, L.; Torres, I.; Uriarte, E.; Y('a)(\~n)ez, M.; Fontenla, J. ?.; Ortuso, F.; Alcaro, S.; Procopio, F.; Borges, F.; Vi(\~n)a, D.
9-fluorenon-4-carboxamides: synthesis, conformational analysis, anti-HSV-2, and immunomodulatory evaluation. Note II
2004-01-01 Arena, A; DI BELLA, R; Neri, S; Ottanà, R; Ortuso, F; Pavone, B; Vigorita, M. G.; Alcaro, S
A chromatographic and computational study on the driving force operating in the exceptionally large enantioseparation of N-thiocarbamoyl-3-(4'-biphenyl)-5-phenyl-4,5-dihydro-(1H) pyrazole on a 4-methylbenzoate cellulose-based chiral stationary phase
2014-01-01 Alcaro, S; Menta, S; Fioravanti, R; Cirilli, R; Ortuso, F
A Comparative Docking Strategy to Identify Polyphenolic Derivatives as Promising Antineoplastic Binders of G-quadruplex DNA c-myc and bcl-2 Sequences
2016-01-01 Costa, G; Rocca, R; Moraca, F; Talarico, C; Romeo, I; Ortuso, F; Artese, A; Alcaro, S
A comparative study of the in vitro inhibitory activity of tacrine-like molecules (Paraquat, MPTP, MPDP and MPP+) on hydrolysis by acetylcholine and butyrylcholine esterases
2004-01-01 Arcone, R.; Alcaro, S; Battaglia, D.; Gallelli, A.; Iannone, M.; Rotiroti, D.; Vecchio, I.; Ortuso, F
A Computational pathway toward the rational design of azinomycin analogues
2008-01-01 Ortuso, F; Pasceri, R; Coleman, R. S.; Artese, A; Alcaro, S
A computer-assisted discovery of novel potential anti-obesity compounds as selective carbonic anhydrase VA inhibitors
2019-01-01 Costa, G.; Carta, F.; Ambrosio, F. A.; Artese, A.; Ortuso, F.; Moraca, F.; Rocca, R.; Romeo, I.; Lupia, A.; Maruca, A.; Bagetta, D.; Catalano, R.; Vullo, D.; Alcaro, S.; Supuran, C. T.
A Dynamic and Effective Peptide-Based Strategy for Promptly Addressing Emerging SARS-CoV-2 Variants of Concern
2024-01-01 Murdocca, M.; Romeo, I.; Citro, G.; Latini, A.; Centofanti, F.; Bugatti, A.; Caccuri, F.; Caruso, A.; Ortuso, F.; Alcaro, S.; Sangiuolo, F.; Novelli, G.
A Fhit-mimetic peptide suppresses annexin A4-mediated chemoresistance to paclitaxel in lung cancer cells
2016-01-01 Gaudio, E; Paduano, F; Ngankeu, A; Ortuso, F; Lovat, F; Pinton, S; D'Agostino, S; Zanesi, N; Aqeilan, Ri; Campiglia, P; Novellino, E; Alcaro, S; Croce, Cm; Trapasso, F
A new series of flavones, thioflavones, and flavanones as selective monoamine oxidase-B inhibitors
2010-01-01 Chimenti, F; Fioravanti, R; Bolasco, A; Chimenti, P; Secci, D; Rossi, F; Yáñez, M; Orallo, F; Alcaro, S; Cirilli, R; Ferretti, R; Sanna, M. L.; Ortuso, F
A Pipeline To Enhance Ligand Virtual Screening: Integrating Molecular Dynamics and Fingerprints for Ligand and Proteins
2015-01-01 Spyrakis, F; Benedetti, P; Decherchi, S; Rocchia, W; Cavalli, A; Ortuso, F; Baroni, M; Cruciani, G; Alcaro, S
An approach to address Candida rugosa lipase regioselectivity in the acylation reactions of trytilated glucosides
2007-01-01 Palocci, C; Falconi, M; Alcaro, S; Tafi, A; Puglisi, R; Botta, M; Alberghina, L; Cernia, E; Ortuso, F
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
"Synthesis, Biological Evaluation and Molecular Modeling of Natural and Semi-synthetic Oleuropeine Drivates as Cox-l and -2 Inhibitors | 1-gen-2008 | Procopio, Antonio; Stefano, Alcaro; Ortuso, Francesco; Nardi, M; Giovanni, Sindona; Paolo, Sacchelta; Oliverio, Manuela | |
(E)-3-Heteroarylidenechroman-4-ones as potent and selective monoamine oxidase-B inhibitors | 1-gen-2016 | Desideri, N; Proietti Monaco, L; Fioravanti, R; Biava, M; Yáñez, M; Ortuso, F; Alcaro, S | |
1,5-Diphenylpenta-2,4-dien-1-ones as potent and selective monoamine oxidase-B inhibitors | 1-gen-2013 | Desideri, N; Fioravanti, R; Proietti Monaco, L; Biava, M; Yáñez, M; Ortuso, F; Alcaro, S | |
1- acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazole; a new scaffold for monoaminoxidase inhibitors: design, synthesis, and biological properties | 1-gen-2008 | Vigo, S; Alcaro, S; Bolasco, A; Cardia, C; Distinto, S; Maccioni, E; Orallo, F; Ortuso, F; Sanna, M. L.; Secci, D; Yanez, M | |
1-benzenesulfonamide-1(H)-pyrazoles and 3-benzenesulfonamide-4-tiazolidinones, two promising scaffolds for the design of cycloxygenase inhibitors | 1-gen-2008 | SANNA M., L; Alcaro, S; Bolasco, A; Cardia, C; Cirilli, R; Distinto, S; Maccioni, E; Orallo, F; Ortuso, F; Secci, D; Vigo, S; Yanez, M | |
4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis | 1-gen-2019 | Secci, D; Carradori, S; Petzer, A; Guglielmi, P; D'Ascenzio, M; Chimenti, P; Bagetta, D; Alcaro, S; Zengin, G; Petzer, Jp; Ortuso, F | |
4-carbossamido-9-fluorenoni: proprietà anti-HSV-2 e immunostimolanti | 1-gen-2004 | Alcaro, S; Arena, A.; DI BELLA, R.; Ortuso, F.; Ottan, R.; Neri, S.; Pavone, B.; Vigorita, M. G. | |
8-Amide and 8-carbamate substitution patterns as modulators of 7-hydroxy-4-methylcoumarin's antidepressant profile: Synthesis, biological evaluation and docking studies | 1-gen-2023 | Matos, M. J.; Novo, P.; Mayan, L.; Torres, I.; Uriarte, E.; Yanez, M.; Fontenla, J. A.; Ortuso, F.; Alcaro, S.; Procopio, F.; Rodriguez-Franco, M. I.; Val, C.; Loza, M. I.; Brea, J.; Borges, F.; Vina, D. | |
8-Amide and 8-Carbamate Substitution Patterns as Modulators of 7-Hydroxy-4-Methylcoumarin{'}s Antidepressant Profile: Synthesis, MAO Inhibition, Cytotoxicity and Docking Studies | 1-gen-2022 | Matos, M. J.; Novo, P.; May('a)n, L.; Torres, I.; Uriarte, E.; Y('a)(\~n)ez, M.; Fontenla, J. ?.; Ortuso, F.; Alcaro, S.; Procopio, F.; Borges, F.; Vi(\~n)a, D. | |
9-fluorenon-4-carboxamides: synthesis, conformational analysis, anti-HSV-2, and immunomodulatory evaluation. Note II | 1-gen-2004 | Arena, A; DI BELLA, R; Neri, S; Ottanà, R; Ortuso, F; Pavone, B; Vigorita, M. G.; Alcaro, S | |
A chromatographic and computational study on the driving force operating in the exceptionally large enantioseparation of N-thiocarbamoyl-3-(4'-biphenyl)-5-phenyl-4,5-dihydro-(1H) pyrazole on a 4-methylbenzoate cellulose-based chiral stationary phase | 1-gen-2014 | Alcaro, S; Menta, S; Fioravanti, R; Cirilli, R; Ortuso, F | |
A Comparative Docking Strategy to Identify Polyphenolic Derivatives as Promising Antineoplastic Binders of G-quadruplex DNA c-myc and bcl-2 Sequences | 1-gen-2016 | Costa, G; Rocca, R; Moraca, F; Talarico, C; Romeo, I; Ortuso, F; Artese, A; Alcaro, S | |
A comparative study of the in vitro inhibitory activity of tacrine-like molecules (Paraquat, MPTP, MPDP and MPP+) on hydrolysis by acetylcholine and butyrylcholine esterases | 1-gen-2004 | Arcone, R.; Alcaro, S; Battaglia, D.; Gallelli, A.; Iannone, M.; Rotiroti, D.; Vecchio, I.; Ortuso, F | |
A Computational pathway toward the rational design of azinomycin analogues | 1-gen-2008 | Ortuso, F; Pasceri, R; Coleman, R. S.; Artese, A; Alcaro, S | |
A computer-assisted discovery of novel potential anti-obesity compounds as selective carbonic anhydrase VA inhibitors | 1-gen-2019 | Costa, G.; Carta, F.; Ambrosio, F. A.; Artese, A.; Ortuso, F.; Moraca, F.; Rocca, R.; Romeo, I.; Lupia, A.; Maruca, A.; Bagetta, D.; Catalano, R.; Vullo, D.; Alcaro, S.; Supuran, C. T. | |
A Dynamic and Effective Peptide-Based Strategy for Promptly Addressing Emerging SARS-CoV-2 Variants of Concern | 1-gen-2024 | Murdocca, M.; Romeo, I.; Citro, G.; Latini, A.; Centofanti, F.; Bugatti, A.; Caccuri, F.; Caruso, A.; Ortuso, F.; Alcaro, S.; Sangiuolo, F.; Novelli, G. | |
A Fhit-mimetic peptide suppresses annexin A4-mediated chemoresistance to paclitaxel in lung cancer cells | 1-gen-2016 | Gaudio, E; Paduano, F; Ngankeu, A; Ortuso, F; Lovat, F; Pinton, S; D'Agostino, S; Zanesi, N; Aqeilan, Ri; Campiglia, P; Novellino, E; Alcaro, S; Croce, Cm; Trapasso, F | |
A new series of flavones, thioflavones, and flavanones as selective monoamine oxidase-B inhibitors | 1-gen-2010 | Chimenti, F; Fioravanti, R; Bolasco, A; Chimenti, P; Secci, D; Rossi, F; Yáñez, M; Orallo, F; Alcaro, S; Cirilli, R; Ferretti, R; Sanna, M. L.; Ortuso, F | |
A Pipeline To Enhance Ligand Virtual Screening: Integrating Molecular Dynamics and Fingerprints for Ligand and Proteins | 1-gen-2015 | Spyrakis, F; Benedetti, P; Decherchi, S; Rocchia, W; Cavalli, A; Ortuso, F; Baroni, M; Cruciani, G; Alcaro, S | |
An approach to address Candida rugosa lipase regioselectivity in the acylation reactions of trytilated glucosides | 1-gen-2007 | Palocci, C; Falconi, M; Alcaro, S; Tafi, A; Puglisi, R; Botta, M; Alberghina, L; Cernia, E; Ortuso, F |