4-Oxoquinolines and monoamine oxidase: When tautomerism matters
2021-01-01 Mesiti, Francesco; Maruca, Annalisa; Silva, Vera; Rocca, Roberta; Fernandes, Carlos; Remião, Fernando; Uriarte, Eugenio; Alcaro, Stefano; Gaspar, Alexandra; Borges, Fernanda
From Nature to Synthetic Compounds: Novel 1(N),2,3 Trisubstituted-5-oxopyrrolidines Targeting Multiple Myeloma Cells
2022-01-01 Listro, Roberta; Malacrida, Alessio; Ambrosio, Francesca Alessandra; Rossino, Giacomo; Di Giacomo, Marcello; Cavalloro, Valeria; Garbagnoli, Martina; Linciano, Pasquale; Rossi, Daniela; Cavaletti, Guido; Costa, Giosuè; Alcaro, Stefano; Miloso, Mariarosaria; Collina, Simona
Targeting SARS-CoV-2 nsp13 Helicase and Assessment of Druggability Pockets: Identification of Two Potent Inhibitors by a Multi-Site In Silico Drug Repurposing Approach
2022-01-01 Romeo, Isabella; Ambrosio, Francesca Alessandra; Costa, Giosuè; Corona, Angela; Alkhatib, Mohammad; Salpini, Romina; Lemme, Saverio; Vergni, Davide; Svicher, Valentina; Santoro, Maria Mercedes; Tramontano, Enzo; Ceccherini-Silberstein, Francesca; Artese, Anna; Alcaro, Stefano
The Tumour Suppressor Fhit Protein Activates C-Raf Ubiquitination and Degradation in Human Melanoma Cells by Interacting with Hsp90
2022-01-01 Paduano, Francesco; Gaudio, Eugenio; Trapasso, Francesco
Evaluation of chromane derivatives: Promising privileged scaffolds for lead discovery within Alzheimer's disease
2022-01-01 Moutayakine, A.; Marques, C.; Lopez, O.; Bagetta, D.; Leitzbach, L.; Hagenow, S.; Carreiro, E. P.; Stark, H.; Alcaro, S.; Fernandez-Bolanos, J. G.; Burke, A. J.
The New Microtubule-Targeting Agent SIX2G Induces Immunogenic Cell Death in Multiple Myeloma
2022-01-01 Grillone, K.; Riillo, C.; Rocca, R.; Ascrizzi, S.; Spano, V.; Scionti, F.; Polera, N.; Maruca, A.; Barreca, M.; Juli, G.; Arbitrio, M.; Di Martino, M. T.; Caracciolo, D.; Tagliaferri, P.; Alcaro, S.; Montalbano, A.; Barraja, P.; Tassone, P.
Design and synthesis of chromone-based monoamine oxidase B inhibitors with improved drug-like properties
2022-01-01 Reis, J.; Fernandes, C.; Salem, H.; Maia, M.; Tome, C.; Benfeito, S.; Teixeira, J.; Oliveira, P. J.; Uriarte, E.; Ortuso, F.; Alcaro, S.; Bagetta, D.; Cagide, F.; Borges, F.
Annona cherimola Mill. Leaf Extracts Affect Melanoma Cells Growth and Progression
2022-01-01 Iacopetta, D.; Fazio, A.; La Torre, C.; Barbarossa, A.; Ceramella, J.; Francomano, F.; Saturnino, C.; El-Kashef, H.; Alcaro, S.; Sinicropi, M. S.
Design, Synthesis, and In Vitro, In Silico and In Cellulo Evaluation of New Pyrimidine and Pyridine Amide and Carbamate Derivatives as Multi-Functional Cholinesterase Inhibitors
2022-01-01 Bortolami, M.; Pandolfi, F.; Tudino, V.; Messore, A.; Madia, V. N.; De Vita, D.; Di Santo, R.; Costi, R.; Romeo, I.; Alcaro, S.; Colone, M.; Stringaro, A.; Espargaro, A.; Sabate, R.; Scipione, L.
Mediterranean Diet: The Beneficial Effects of Lycopene in Non-Alcoholic Fatty Liver Disease
2022-01-01 Abenavoli, L.; Procopio, A. C.; Paravati, M. R.; Costa, G.; Milic, N.; Alcaro, S.; Luzza, F.
Transcriptome and computational analysis assess the anti-tubulin activity of [1,2]oxazole derivatives in lymphoma
2022-01-01 Barreca, M.; Spanò, V.; Rocca, R.; Bivacqua, R.; Maruca, A.; Montalbano, A.; Raimondi, M. V.; Tarantelli, C.; Gaudio, E.; Cascione, L.; Rinaldi, A.; Bai, R.; Prota, A.; Abel, A. C.; Steinmetz, M.; Alcaro, S.; Hamel, E.; Bertoni, F.; Barraja, P.
Exploiting DNA Ligase III addiction of multiple myeloma by flavonoid Rhamnetin
2022-01-01 Caracciolo, Daniele; Juli, Giada; Riillo, Caterina; Coricello, Adriana; Vasile, Francesca; Pollastri, Sara; Rocca, Roberta; Scionti, Francesca; Polerà, Nicoletta; Grillone, Katia; Arbitrio, Mariamena; Staropoli, Nicoletta; Caparello, Basilio; Britti, Domenico; Loprete, Giovanni; Costa, Giosuè; Di Martino, Maria Teresa; Alcaro, Stefano; Tagliaferri, Pierosandro; Tassone, Pierfrancesco
Development of [1,2]oxazoloisoindoles tubulin polymerization inhibitors: Further chemical modifications and potential therapeutic effects against lymphomas
2022-01-01 Barreca, Marilia; Spanò, Virginia; Rocca, Roberta; Bivacqua, Roberta; Abel, Anne-Catherine; Maruca, Annalisa; Montalbano, Alessandra; Raimondi, Maria Valeria; Tarantelli, Chiara; Gaudio, Eugenio; Cascione, Luciano; Rinaldi, Andrea; Bai, Ruoli; Steinmetz, Michel O.; Prota, Andrea E.; Alcaro, Stefano; Hamel, Ernest; Bertoni, Francesco; Barraja, Paola
Formulation of Solid Lipid Nanoparticles Loaded with Nociceptin/Orphanin FQ (N/OFQ) and Characterization in a Murine Model of Airway Hyperresponsiveness
2022-01-01 Mirra, D.; Spaziano, G.; Esposito, R.; Santonocito, D.; Filosa, R.; Roviezzo, F.; Malgieri, G.; D'Abrosca, G.; Iovino, P.; Gallelli, L.; Fattorusso, R.; Puglia, C.; D'Agostino, B.
Synthesis of 2H-Imidazo[2′,1':2,3] [1,3]thiazolo[4,5-e]isoindol-8-yl-phenylureas with promising therapeutic features for the treatment of acute myeloid leukemia (AML) with FLT3/ITD mutations
2022-01-01 Cilibrasi, V.; Spano, V.; Bortolozzi, R.; Barreca, M.; Raimondi, M. V.; Rocca, R.; Maruca, A.; Montalbano, A.; Alcaro, S.; Ronca, R.; Viola, G.; Barraja, P.
Riluzole-Rasagiline Hybrids: Toward the Development of Multi-Target-Directed Ligands for Amyotrophic Lateral Sclerosis
2022-01-01 Albertini, Claudia; Salerno, Alessandra; Atzeni, Silvia; Uliassi, Elisa; Massenzio, Francesca; Maruca, Annalisa; Rocca, Roberta; Mecava, Marko; Silva, Filomena S G; Mena, Débora; Valente, Pedro; Duarte, Ana I; Chavarria, Daniel; Bissaro, Maicol; Moro, Stefano; Federico, Stephanie; Spalluto, Giampiero; Soukup, Ondřej; Borges, Fernanda; Alcaro, Stefano; Monti, Barbara; Oliveira, Paulo J; Menéndez, Josè C; Bolognesi, Maria Laura
Non-uniform Self-folding of Helical Poly(fluorenevinylene) Derivatives in the Solid State Leading to Amplified Circular Dichroism and Circularly Polarized Light Emission
2022-01-01 Wu, P.; Pietropaolo, A.; Fortino, M.; Shimoda, S.; Maeda, K.; Nishimura, T.; Bando, M.; Naga, N.; Nakano, T.
Optimal acquisition time window and simplified quantification of dopamine transporter availability using 18F-FE-PE2I in healthy controls and Parkinson's disease patients.
2016-01-01 Sonni, I; Fazio, P; Schain, M; Halldin, C; Svenningsson, P; Farde, L; Varrone, A
An 8-week open label trial of L-Threonic Acid Magnesium Salt in patients with mild to moderate dementia
2017-01-01 Wroolie, Te; Chen, K; Watson, Kt; Iagaru, A; Sonni, I; Snyder, N; Lee, W; Reiman, Em; Rasgon, Nl
Prospective Evaluation of 68Ga-RM2 PET/MRI in Patients with Biochemical Recurrence of Prostate Cancer and Negative Conventional Imaging
2018-01-01 Minamimoto, R; Sonni, I; Hancock, S; Vasanawala, S; Loening, A; Gambhir, Ss; Iagaru, A
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 4-Oxoquinolines and monoamine oxidase: When tautomerism matters | 1-gen-2021 | Mesiti, Francesco; Maruca, Annalisa; Silva, Vera; Rocca, Roberta; Fernandes, Carlos; Remião, Fernando; Uriarte, Eugenio; Alcaro, Stefano; Gaspar, Alexandra; Borges, Fernanda | |
| From Nature to Synthetic Compounds: Novel 1(N),2,3 Trisubstituted-5-oxopyrrolidines Targeting Multiple Myeloma Cells | 1-gen-2022 | Listro, Roberta; Malacrida, Alessio; Ambrosio, Francesca Alessandra; Rossino, Giacomo; Di Giacomo, Marcello; Cavalloro, Valeria; Garbagnoli, Martina; Linciano, Pasquale; Rossi, Daniela; Cavaletti, Guido; Costa, Giosuè; Alcaro, Stefano; Miloso, Mariarosaria; Collina, Simona | |
| Targeting SARS-CoV-2 nsp13 Helicase and Assessment of Druggability Pockets: Identification of Two Potent Inhibitors by a Multi-Site In Silico Drug Repurposing Approach | 1-gen-2022 | Romeo, Isabella; Ambrosio, Francesca Alessandra; Costa, Giosuè; Corona, Angela; Alkhatib, Mohammad; Salpini, Romina; Lemme, Saverio; Vergni, Davide; Svicher, Valentina; Santoro, Maria Mercedes; Tramontano, Enzo; Ceccherini-Silberstein, Francesca; Artese, Anna; Alcaro, Stefano | |
| The Tumour Suppressor Fhit Protein Activates C-Raf Ubiquitination and Degradation in Human Melanoma Cells by Interacting with Hsp90 | 1-gen-2022 | Paduano, Francesco; Gaudio, Eugenio; Trapasso, Francesco | |
| Evaluation of chromane derivatives: Promising privileged scaffolds for lead discovery within Alzheimer's disease | 1-gen-2022 | Moutayakine, A.; Marques, C.; Lopez, O.; Bagetta, D.; Leitzbach, L.; Hagenow, S.; Carreiro, E. P.; Stark, H.; Alcaro, S.; Fernandez-Bolanos, J. G.; Burke, A. J. | |
| The New Microtubule-Targeting Agent SIX2G Induces Immunogenic Cell Death in Multiple Myeloma | 1-gen-2022 | Grillone, K.; Riillo, C.; Rocca, R.; Ascrizzi, S.; Spano, V.; Scionti, F.; Polera, N.; Maruca, A.; Barreca, M.; Juli, G.; Arbitrio, M.; Di Martino, M. T.; Caracciolo, D.; Tagliaferri, P.; Alcaro, S.; Montalbano, A.; Barraja, P.; Tassone, P. | |
| Design and synthesis of chromone-based monoamine oxidase B inhibitors with improved drug-like properties | 1-gen-2022 | Reis, J.; Fernandes, C.; Salem, H.; Maia, M.; Tome, C.; Benfeito, S.; Teixeira, J.; Oliveira, P. J.; Uriarte, E.; Ortuso, F.; Alcaro, S.; Bagetta, D.; Cagide, F.; Borges, F. | |
| Annona cherimola Mill. Leaf Extracts Affect Melanoma Cells Growth and Progression | 1-gen-2022 | Iacopetta, D.; Fazio, A.; La Torre, C.; Barbarossa, A.; Ceramella, J.; Francomano, F.; Saturnino, C.; El-Kashef, H.; Alcaro, S.; Sinicropi, M. S. | |
| Design, Synthesis, and In Vitro, In Silico and In Cellulo Evaluation of New Pyrimidine and Pyridine Amide and Carbamate Derivatives as Multi-Functional Cholinesterase Inhibitors | 1-gen-2022 | Bortolami, M.; Pandolfi, F.; Tudino, V.; Messore, A.; Madia, V. N.; De Vita, D.; Di Santo, R.; Costi, R.; Romeo, I.; Alcaro, S.; Colone, M.; Stringaro, A.; Espargaro, A.; Sabate, R.; Scipione, L. | |
| Mediterranean Diet: The Beneficial Effects of Lycopene in Non-Alcoholic Fatty Liver Disease | 1-gen-2022 | Abenavoli, L.; Procopio, A. C.; Paravati, M. R.; Costa, G.; Milic, N.; Alcaro, S.; Luzza, F. | |
| Transcriptome and computational analysis assess the anti-tubulin activity of [1,2]oxazole derivatives in lymphoma | 1-gen-2022 | Barreca, M.; Spanò, V.; Rocca, R.; Bivacqua, R.; Maruca, A.; Montalbano, A.; Raimondi, M. V.; Tarantelli, C.; Gaudio, E.; Cascione, L.; Rinaldi, A.; Bai, R.; Prota, A.; Abel, A. C.; Steinmetz, M.; Alcaro, S.; Hamel, E.; Bertoni, F.; Barraja, P. | |
| Exploiting DNA Ligase III addiction of multiple myeloma by flavonoid Rhamnetin | 1-gen-2022 | Caracciolo, Daniele; Juli, Giada; Riillo, Caterina; Coricello, Adriana; Vasile, Francesca; Pollastri, Sara; Rocca, Roberta; Scionti, Francesca; Polerà, Nicoletta; Grillone, Katia; Arbitrio, Mariamena; Staropoli, Nicoletta; Caparello, Basilio; Britti, Domenico; Loprete, Giovanni; Costa, Giosuè; Di Martino, Maria Teresa; Alcaro, Stefano; Tagliaferri, Pierosandro; Tassone, Pierfrancesco | |
| Development of [1,2]oxazoloisoindoles tubulin polymerization inhibitors: Further chemical modifications and potential therapeutic effects against lymphomas | 1-gen-2022 | Barreca, Marilia; Spanò, Virginia; Rocca, Roberta; Bivacqua, Roberta; Abel, Anne-Catherine; Maruca, Annalisa; Montalbano, Alessandra; Raimondi, Maria Valeria; Tarantelli, Chiara; Gaudio, Eugenio; Cascione, Luciano; Rinaldi, Andrea; Bai, Ruoli; Steinmetz, Michel O.; Prota, Andrea E.; Alcaro, Stefano; Hamel, Ernest; Bertoni, Francesco; Barraja, Paola | |
| Formulation of Solid Lipid Nanoparticles Loaded with Nociceptin/Orphanin FQ (N/OFQ) and Characterization in a Murine Model of Airway Hyperresponsiveness | 1-gen-2022 | Mirra, D.; Spaziano, G.; Esposito, R.; Santonocito, D.; Filosa, R.; Roviezzo, F.; Malgieri, G.; D'Abrosca, G.; Iovino, P.; Gallelli, L.; Fattorusso, R.; Puglia, C.; D'Agostino, B. | |
| Synthesis of 2H-Imidazo[2′,1':2,3] [1,3]thiazolo[4,5-e]isoindol-8-yl-phenylureas with promising therapeutic features for the treatment of acute myeloid leukemia (AML) with FLT3/ITD mutations | 1-gen-2022 | Cilibrasi, V.; Spano, V.; Bortolozzi, R.; Barreca, M.; Raimondi, M. V.; Rocca, R.; Maruca, A.; Montalbano, A.; Alcaro, S.; Ronca, R.; Viola, G.; Barraja, P. | |
| Riluzole-Rasagiline Hybrids: Toward the Development of Multi-Target-Directed Ligands for Amyotrophic Lateral Sclerosis | 1-gen-2022 | Albertini, Claudia; Salerno, Alessandra; Atzeni, Silvia; Uliassi, Elisa; Massenzio, Francesca; Maruca, Annalisa; Rocca, Roberta; Mecava, Marko; Silva, Filomena S G; Mena, Débora; Valente, Pedro; Duarte, Ana I; Chavarria, Daniel; Bissaro, Maicol; Moro, Stefano; Federico, Stephanie; Spalluto, Giampiero; Soukup, Ondřej; Borges, Fernanda; Alcaro, Stefano; Monti, Barbara; Oliveira, Paulo J; Menéndez, Josè C; Bolognesi, Maria Laura | |
| Non-uniform Self-folding of Helical Poly(fluorenevinylene) Derivatives in the Solid State Leading to Amplified Circular Dichroism and Circularly Polarized Light Emission | 1-gen-2022 | Wu, P.; Pietropaolo, A.; Fortino, M.; Shimoda, S.; Maeda, K.; Nishimura, T.; Bando, M.; Naga, N.; Nakano, T. | |
| Optimal acquisition time window and simplified quantification of dopamine transporter availability using 18F-FE-PE2I in healthy controls and Parkinson's disease patients. | 1-gen-2016 | Sonni, I; Fazio, P; Schain, M; Halldin, C; Svenningsson, P; Farde, L; Varrone, A | |
| An 8-week open label trial of L-Threonic Acid Magnesium Salt in patients with mild to moderate dementia | 1-gen-2017 | Wroolie, Te; Chen, K; Watson, Kt; Iagaru, A; Sonni, I; Snyder, N; Lee, W; Reiman, Em; Rasgon, Nl | |
| Prospective Evaluation of 68Ga-RM2 PET/MRI in Patients with Biochemical Recurrence of Prostate Cancer and Negative Conventional Imaging | 1-gen-2018 | Minamimoto, R; Sonni, I; Hancock, S; Vasanawala, S; Loening, A; Gambhir, Ss; Iagaru, A |
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