Sfoglia per Rivista BIOORGANIC
Design and synthesis of DNA-intercalating 9-fluoren-β-O-glycosides as potential IFN-inducers, and antiviral and cytostatic agents
2004-01-01 Arena, A; Neri, S; Ottanà, R; Ortuso, F; Pavone, B; Vigorita, M. G.; Alcaro, S
Design of 1-substituted 2-arylmethyl-4,5-methylenedioxybenzene derivatives as antiseizure agents
2004-01-01 Micale, N; De Sarro, G; Ferreri, G; Zappala, M; Grasso, S; Puia, G; De Micheli, C
Design, synthesis, and SAR analysis of novel selective sigma(1) ligands
2007-01-01 Collina, S; Loddo, G; Urbano, M; Linati, L; Callegari, A; Ortuso, F; Laggner, C; Langer, T; Prezzavento, O; Ronsisvalle, G; Azzolina, O; Alcaro, S
Design, synthesis, biophysical and biological studies of trisubstituted naphthalimides as G-quadruplex ligands
2011-01-01 Peduto, A; Pagano, B; Petronzi, C; Massa, A; Esposito, V; Virgilio, A; Paduano, F; Trapasso, F; Fiorito, F; Florio, S; Giancola, C; Galeone, A; Filosa, R
Development of 3-substituted-1H-indole derivatives as NR2B/NMDA receptor antagonists
2009-01-01 Gitto, R; Luca, Ld; Ferro, S; Citraro, R; Sarro, Gd; Costa, L; Ciranna, L; Chimirri, A
Evaluation of chromane derivatives: Promising privileged scaffolds for lead discovery within Alzheimer's disease
2022-01-01 Moutayakine, A.; Marques, C.; Lopez, O.; Bagetta, D.; Leitzbach, L.; Hagenow, S.; Carreiro, E. P.; Stark, H.; Alcaro, S.; Fernandez-Bolanos, J. G.; Burke, A. J.
Exploring new chemical functionalities to improve aromatase inhibition of steroids
2016-01-01 Varela, Cl; Amaral, C; Correia-da-Silva, G; Costa, Sc; Carvalho, Ra; Costa, G; Alcaro, S; Teixeira, Naa; Tavares-da-Silva, Ej; Roleira, Fmf
Identification of the stereochemical requirements in the 4-aryl-2-cycloalkylidenhydrazinylthiazole scaffold for the design of selective human monoamine oxidase B inhibitors.
2014-01-01 D'Ascenzio, M; Carradori, S; Secci, D; Mannina, L; Sobolev, Ap; De Monte, C; Cirilli, R; Yáñez, M; Ortuso, F; Alcaro, S
Investigations on the 2-thiazolylhydrazyne scaffold: synthesis and molecular modeling of selective human monoamine oxidase inhibitors
2010-01-01 Chimenti, F; Bolasco, A; Secci, D; Chimenti, P; Granese, A; Carradori, S; Yáñez, M; Orallo, F; Alcaro, S; Ortuso, F
Macrocyclic naphthalene diimides as G-quadruplex binders.
2015-01-01 Marchetti, C; Minarini, A; Tumiatti, V; Moraca, F; Parrotta, L; Alcaro, S; Rigo, R; Sissi, C; Gunaratnam, M; Ohnmacht, Sa; Neidle, S; Milelli, A.
N-Alkyl dien- and trienamides from the roots of Otanthus maritimus with binding affinity for opioid and cannabinoid receptors.
2013-01-01 Ruiu, S; Anzani, N; Orrù, A; Floris, C; Caboni, P; Maccioni, E; Distinto, S; Alcaro, S; Cottiglia, F.
Structure-activity relationships of 2-aryl-2,5-dihydropyridazino[4,3-b]indol-3(3H)-ones at the benzodiazepine receptor
1996-01-01 Palluotto, F; Carotti, A; Casini, G; Campagna, F; Genchi, G; Rizzo, M; De Sarro, G
Structure-guided design of new indoles as negative allosteric modulators (NAMs) of N-methyl-D-aspartate receptor (NMDAR) containing GluN2B subunit
2016-01-01 Buemi, Mr; De Luca, L; Ferro, S; Russo, E; Gitto, R; De Sarro, G
Synthesis and anticonvulsant evaluation of N-substituted isoquinoline AMPA receptor antagonists
2008-01-01 Gitto, R; DE LUCA, L; Pagano, B; Citraro, R; DE SARRO, G; Costa, L; Ciranna, L; Chimirri, A
Synthesis and evaluation of pharmacological pro. le of 1-aryl-6,7-dimethoxy-3,4-dihydroisoquinoline-2(1H)-sulfonamides
2009-01-01 Gitto, R; Ferro, S; Agnello, S; De Luca, L; De Sarro, G; Vullo, D; Supuran, Ct; Chimirri, A; Russo, E
Synthesis, modelling and biological characterization of 3-substituted-1H-indoles as ligands of GluN2B-containing N-methyl-d-aspartate receptors
2014-01-01 Gitto, R; De Luca, L; Ferro, S; Russo, E; De Sarro, G; Chisari, M; Ciranna, L; Alvarez-Builla, J; Alajarin, R; Buemi, Mr; Chimirri, A
Synthesis, resolution, stereochemistry, and molecular modeling of (R)- and (S)-2-acetyl-1-(4 '-chlorophenyl)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline AMPAR antagonists
2007-01-01 Gitto, R; Ficarra, R; Stancanelli, R; Guardo, M; De Luca, L; Barreca, Ml; Pagano, B; Rotondo, A; Bruno, G; Russo, E; Chimirri, A; De Sarro, G
Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitors
2010-01-01 Chimenti, F; Secci, D; Bolasco, A; Chimenti, P; Granese, A; Carradori, S; Maccioni, E; Cardia, M. C.; Yáñez, M; Orallo, F; Alcaro, S; Cirilli, R; Ferretti, R; Distinto, S; Kirchmair, J; Langer, T; Ortuso, F
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Design and synthesis of DNA-intercalating 9-fluoren-β-O-glycosides as potential IFN-inducers, and antiviral and cytostatic agents | 1-gen-2004 | Arena, A; Neri, S; Ottanà, R; Ortuso, F; Pavone, B; Vigorita, M. G.; Alcaro, S | |
Design of 1-substituted 2-arylmethyl-4,5-methylenedioxybenzene derivatives as antiseizure agents | 1-gen-2004 | Micale, N; De Sarro, G; Ferreri, G; Zappala, M; Grasso, S; Puia, G; De Micheli, C | |
Design, synthesis, and SAR analysis of novel selective sigma(1) ligands | 1-gen-2007 | Collina, S; Loddo, G; Urbano, M; Linati, L; Callegari, A; Ortuso, F; Laggner, C; Langer, T; Prezzavento, O; Ronsisvalle, G; Azzolina, O; Alcaro, S | |
Design, synthesis, biophysical and biological studies of trisubstituted naphthalimides as G-quadruplex ligands | 1-gen-2011 | Peduto, A; Pagano, B; Petronzi, C; Massa, A; Esposito, V; Virgilio, A; Paduano, F; Trapasso, F; Fiorito, F; Florio, S; Giancola, C; Galeone, A; Filosa, R | |
Development of 3-substituted-1H-indole derivatives as NR2B/NMDA receptor antagonists | 1-gen-2009 | Gitto, R; Luca, Ld; Ferro, S; Citraro, R; Sarro, Gd; Costa, L; Ciranna, L; Chimirri, A | |
Evaluation of chromane derivatives: Promising privileged scaffolds for lead discovery within Alzheimer's disease | 1-gen-2022 | Moutayakine, A.; Marques, C.; Lopez, O.; Bagetta, D.; Leitzbach, L.; Hagenow, S.; Carreiro, E. P.; Stark, H.; Alcaro, S.; Fernandez-Bolanos, J. G.; Burke, A. J. | |
Exploring new chemical functionalities to improve aromatase inhibition of steroids | 1-gen-2016 | Varela, Cl; Amaral, C; Correia-da-Silva, G; Costa, Sc; Carvalho, Ra; Costa, G; Alcaro, S; Teixeira, Naa; Tavares-da-Silva, Ej; Roleira, Fmf | |
Identification of the stereochemical requirements in the 4-aryl-2-cycloalkylidenhydrazinylthiazole scaffold for the design of selective human monoamine oxidase B inhibitors. | 1-gen-2014 | D'Ascenzio, M; Carradori, S; Secci, D; Mannina, L; Sobolev, Ap; De Monte, C; Cirilli, R; Yáñez, M; Ortuso, F; Alcaro, S | |
Investigations on the 2-thiazolylhydrazyne scaffold: synthesis and molecular modeling of selective human monoamine oxidase inhibitors | 1-gen-2010 | Chimenti, F; Bolasco, A; Secci, D; Chimenti, P; Granese, A; Carradori, S; Yáñez, M; Orallo, F; Alcaro, S; Ortuso, F | |
Macrocyclic naphthalene diimides as G-quadruplex binders. | 1-gen-2015 | Marchetti, C; Minarini, A; Tumiatti, V; Moraca, F; Parrotta, L; Alcaro, S; Rigo, R; Sissi, C; Gunaratnam, M; Ohnmacht, Sa; Neidle, S; Milelli, A. | |
N-Alkyl dien- and trienamides from the roots of Otanthus maritimus with binding affinity for opioid and cannabinoid receptors. | 1-gen-2013 | Ruiu, S; Anzani, N; Orrù, A; Floris, C; Caboni, P; Maccioni, E; Distinto, S; Alcaro, S; Cottiglia, F. | |
Structure-activity relationships of 2-aryl-2,5-dihydropyridazino[4,3-b]indol-3(3H)-ones at the benzodiazepine receptor | 1-gen-1996 | Palluotto, F; Carotti, A; Casini, G; Campagna, F; Genchi, G; Rizzo, M; De Sarro, G | |
Structure-guided design of new indoles as negative allosteric modulators (NAMs) of N-methyl-D-aspartate receptor (NMDAR) containing GluN2B subunit | 1-gen-2016 | Buemi, Mr; De Luca, L; Ferro, S; Russo, E; Gitto, R; De Sarro, G | |
Synthesis and anticonvulsant evaluation of N-substituted isoquinoline AMPA receptor antagonists | 1-gen-2008 | Gitto, R; DE LUCA, L; Pagano, B; Citraro, R; DE SARRO, G; Costa, L; Ciranna, L; Chimirri, A | |
Synthesis and evaluation of pharmacological pro. le of 1-aryl-6,7-dimethoxy-3,4-dihydroisoquinoline-2(1H)-sulfonamides | 1-gen-2009 | Gitto, R; Ferro, S; Agnello, S; De Luca, L; De Sarro, G; Vullo, D; Supuran, Ct; Chimirri, A; Russo, E | |
Synthesis, modelling and biological characterization of 3-substituted-1H-indoles as ligands of GluN2B-containing N-methyl-d-aspartate receptors | 1-gen-2014 | Gitto, R; De Luca, L; Ferro, S; Russo, E; De Sarro, G; Chisari, M; Ciranna, L; Alvarez-Builla, J; Alajarin, R; Buemi, Mr; Chimirri, A | |
Synthesis, resolution, stereochemistry, and molecular modeling of (R)- and (S)-2-acetyl-1-(4 '-chlorophenyl)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline AMPAR antagonists | 1-gen-2007 | Gitto, R; Ficarra, R; Stancanelli, R; Guardo, M; De Luca, L; Barreca, Ml; Pagano, B; Rotondo, A; Bruno, G; Russo, E; Chimirri, A; De Sarro, G | |
Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitors | 1-gen-2010 | Chimenti, F; Secci, D; Bolasco, A; Chimenti, P; Granese, A; Carradori, S; Maccioni, E; Cardia, M. C.; Yáñez, M; Orallo, F; Alcaro, S; Cirilli, R; Ferretti, R; Distinto, S; Kirchmair, J; Langer, T; Ortuso, F |
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