Sfoglia per Rivista BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
1-Aryl-6,7-methylenedioxy-3H-quinazolin-4-ones as anticonvulsant agents
2003-01-01 Zappala, M; Grasso, S; Micale, N; Zuccala, G; Menniti, Fs; Ferreri, G; De Sarro, G; De Micheli, C
Chiral 3,3'-(1,2-ethanediyl)-bis[2-(3,4-dimethoxyphenyl)-4-thiazolidinones] with anti-inflammatory activity. part II: evaluation of cox-2 selectivity and modelling
2003-01-01 Vigorita, M. G.; Ottana, R; Monforte, F; Maccari, R; Monforte, M. T.; Trovato, A; Taviano, M. F.; Miceli, N; DE LUCA, G; Ortuso, F; Alcaro, S
Chiral arylpyrrolidinols: preparation and biological profile
2005-01-01 Collina, S.; Rossi, D.; Loddo, G.; Barbieri, A.; Lanza, E.; Linati, L.; Alcaro, S; Gallelli, A.; Azzolina, O.; Ghislandi, V.
Chromone-2- and -3-carboxylic acids inhibit differently monoamine oxidases A and B
2010-01-01 Alcaro, S; Gaspar, A; Milhazes, N; Orallo, F; Uriarte, E; Yãnez, M; Borges, F; Ortuso, F
Conformational search of antisense nucleotides
2001-01-01 Alcaro, S; Tafi, A.; Wozniak, L. A.; GÁCS-BAITZ, E.; Botta, M.; Ortuso, F
FFAR1/GPR40: One target, different binding sites, many agonists, no drugs, but a continuous and unprofitable tug-of-war between ligand lipophilicity, activity, and toxicity
2021-01-01 Governa, P.; Caroleo, M. C.; Carullo, G.; Aiello, F.; Cione, E.; Manetti, F.
Inhibition of Amine Oxidases Activity by 1-Acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole Derivatives
2002-01-01 Manna, F.; Chimenti, F.; Bolasco, A.; Secci, D.; Bizzarri, B.; Befani, L.; Turini, P.; Mondovi`, B.; Alcaro, S; Tafi, A.
Inhibition of monoamine oxidases by coumarin-3-acyl derivatives: biological activity and computational study
2004-01-01 Chimenti, F.; Secci, D.; Bolasco, A.; Chimenti, P.; Granese, A.; Befani, O.; Turini, P.; Alcaro, S; Ortuso, F
Molecular modeling and enzymatic studies of the interaction of a choline analogue and acetylcholinesterase
2002-01-01 Scipione, L; Ortuso, F; Posca, S; Rispoli, V; Rotiroti, D; Alcaro, S
New 4-[(3-cyclohexyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzene-1-sulfonamides, synthesis and inhibitory activity toward carbonic anhydrase I, II, IX, XII
2015-01-01 Meleddu, R; Maccioni, E; Distinto, S; Bianco, G; Melis, C; Alcaro, S; Cottiglia, F; Ceruso, M; Supuran, Ct
New 7,8-ethylenedioxy-2,3-benzodiazepines as noncompetitive AMPA receptor antagonists
2006-01-01 Zappala, M; Pellicano, A; Micale, N; Menniti, Fs; Ferreri, G; De Sarro, G; Grasso, S; De Micheli, C
New conformationally locked bicyclic N,O-nucleoside analogues of antiviral drugs
2005-01-01 Procopio, A; DE NINO, A; Maiuolo, L; Ortuso, F; Sindona, G; Alcaro, S
Preparation, characterization,molecular modeling and in vitro activity of paclitaxel cyclodextrin complexes
2002-01-01 Ventura, C. A.; Battaglia, D; Ortuso, F; Cattel, L; Puglisi, G; Alcaro, S; Fresta, M; Paolino, D
Quercetin-3-oleoyl derivatives as new GPR40 agonists: Molecular docking studies and functional evaluation
2019-01-01 Carullo, Gabriele; Perri, Mariarita; Manetti, Fabrizio; Aiello, Francesca; Caroleo, Maria Cristina; Cione, Erika
Synthesis and molecular modelling studies of prenylated pyrazolines as MAO-B inhibitors
2010-01-01 Fioravanti, R; Bolasco, A; Manna, F; Rossi, F; Orallo, F; Yáñez, M; Vitali, A; Alcaro, S; Ortuso, F
Synthesis, molecular modeling studies, and selective inhibitory activity against monoamine oxidase of N,N'-bis[2-oxo-2H-benzopyran]-3-carboxamides
2006-01-01 Chimenti, F; Secci, D; Bolasco, A; Chimenti, P; Granese, A; Carradori, S; Befani, O; Turini, P; Ortuso, F; Alcaro, S
Tetraplex DNA specific ligands based on the fluorenone-carboxamide scaffold
2007-01-01 Alcaro, S; Artese, A; Iley, J. N.; Maccari, R; Missailidis, S; Ottana, R; Ragazzon, P; Vigorita, M. G.; Ortuso, F
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 1-Aryl-6,7-methylenedioxy-3H-quinazolin-4-ones as anticonvulsant agents | 1-gen-2003 | Zappala, M; Grasso, S; Micale, N; Zuccala, G; Menniti, Fs; Ferreri, G; De Sarro, G; De Micheli, C | |
| Chiral 3,3'-(1,2-ethanediyl)-bis[2-(3,4-dimethoxyphenyl)-4-thiazolidinones] with anti-inflammatory activity. part II: evaluation of cox-2 selectivity and modelling | 1-gen-2003 | Vigorita, M. G.; Ottana, R; Monforte, F; Maccari, R; Monforte, M. T.; Trovato, A; Taviano, M. F.; Miceli, N; DE LUCA, G; Ortuso, F; Alcaro, S | |
| Chiral arylpyrrolidinols: preparation and biological profile | 1-gen-2005 | Collina, S.; Rossi, D.; Loddo, G.; Barbieri, A.; Lanza, E.; Linati, L.; Alcaro, S; Gallelli, A.; Azzolina, O.; Ghislandi, V. | |
| Chromone-2- and -3-carboxylic acids inhibit differently monoamine oxidases A and B | 1-gen-2010 | Alcaro, S; Gaspar, A; Milhazes, N; Orallo, F; Uriarte, E; Yãnez, M; Borges, F; Ortuso, F | |
| Conformational search of antisense nucleotides | 1-gen-2001 | Alcaro, S; Tafi, A.; Wozniak, L. A.; GÁCS-BAITZ, E.; Botta, M.; Ortuso, F | |
| FFAR1/GPR40: One target, different binding sites, many agonists, no drugs, but a continuous and unprofitable tug-of-war between ligand lipophilicity, activity, and toxicity | 1-gen-2021 | Governa, P.; Caroleo, M. C.; Carullo, G.; Aiello, F.; Cione, E.; Manetti, F. | |
| Inhibition of Amine Oxidases Activity by 1-Acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole Derivatives | 1-gen-2002 | Manna, F.; Chimenti, F.; Bolasco, A.; Secci, D.; Bizzarri, B.; Befani, L.; Turini, P.; Mondovi`, B.; Alcaro, S; Tafi, A. | |
| Inhibition of monoamine oxidases by coumarin-3-acyl derivatives: biological activity and computational study | 1-gen-2004 | Chimenti, F.; Secci, D.; Bolasco, A.; Chimenti, P.; Granese, A.; Befani, O.; Turini, P.; Alcaro, S; Ortuso, F | |
| Molecular modeling and enzymatic studies of the interaction of a choline analogue and acetylcholinesterase | 1-gen-2002 | Scipione, L; Ortuso, F; Posca, S; Rispoli, V; Rotiroti, D; Alcaro, S | |
| New 4-[(3-cyclohexyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzene-1-sulfonamides, synthesis and inhibitory activity toward carbonic anhydrase I, II, IX, XII | 1-gen-2015 | Meleddu, R; Maccioni, E; Distinto, S; Bianco, G; Melis, C; Alcaro, S; Cottiglia, F; Ceruso, M; Supuran, Ct | |
| New 7,8-ethylenedioxy-2,3-benzodiazepines as noncompetitive AMPA receptor antagonists | 1-gen-2006 | Zappala, M; Pellicano, A; Micale, N; Menniti, Fs; Ferreri, G; De Sarro, G; Grasso, S; De Micheli, C | |
| New conformationally locked bicyclic N,O-nucleoside analogues of antiviral drugs | 1-gen-2005 | Procopio, A; DE NINO, A; Maiuolo, L; Ortuso, F; Sindona, G; Alcaro, S | |
| Preparation, characterization,molecular modeling and in vitro activity of paclitaxel cyclodextrin complexes | 1-gen-2002 | Ventura, C. A.; Battaglia, D; Ortuso, F; Cattel, L; Puglisi, G; Alcaro, S; Fresta, M; Paolino, D | |
| Quercetin-3-oleoyl derivatives as new GPR40 agonists: Molecular docking studies and functional evaluation | 1-gen-2019 | Carullo, Gabriele; Perri, Mariarita; Manetti, Fabrizio; Aiello, Francesca; Caroleo, Maria Cristina; Cione, Erika | |
| Synthesis and molecular modelling studies of prenylated pyrazolines as MAO-B inhibitors | 1-gen-2010 | Fioravanti, R; Bolasco, A; Manna, F; Rossi, F; Orallo, F; Yáñez, M; Vitali, A; Alcaro, S; Ortuso, F | |
| Synthesis, molecular modeling studies, and selective inhibitory activity against monoamine oxidase of N,N'-bis[2-oxo-2H-benzopyran]-3-carboxamides | 1-gen-2006 | Chimenti, F; Secci, D; Bolasco, A; Chimenti, P; Granese, A; Carradori, S; Befani, O; Turini, P; Ortuso, F; Alcaro, S | |
| Tetraplex DNA specific ligands based on the fluorenone-carboxamide scaffold | 1-gen-2007 | Alcaro, S; Artese, A; Iley, J. N.; Maccari, R; Missailidis, S; Ottana, R; Ragazzon, P; Vigorita, M. G.; Ortuso, F |
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