Sfoglia per Rivista BIOORGANIC & MEDICINAL CHEMISTRY
2-Aryl-2,5-dihydropyridazino[4,3-b]indol-3(3H)-ones: novel rigid planar benzodiazepine receptor ligands.
1993-01-01 Campagna, F; Carotti, A; Casini, G; Palluotto, F; Genchi, G; De Sarro, G
A new series of flavones, thioflavones, and flavanones as selective monoamine oxidase-B inhibitors
2010-01-01 Chimenti, F; Fioravanti, R; Bolasco, A; Chimenti, P; Secci, D; Rossi, F; Yáñez, M; Orallo, F; Alcaro, S; Cirilli, R; Ferretti, R; Sanna, M. L.; Ortuso, F
Biocatalysed synthesis of β-O-glucosides from 9-fluorenon-2-carbohydroxyesters. Part 3: IFN-inducing and anti-HSV-2 properties
2005-01-01 Arena, A; DI BELLA, R; Neri, S; Ottanà, R; Ortuso, F; Pavone, B; Trincone, A; Vigorita, M. G.; Alcaro, S
Combined NMR-crystallographic and modelling investigation of the inclusion of molsidomine into alpha-, beta- and gamma-cyclodextrins
2005-01-01 Uccello-Barretta, G; Balzano, F; Paolino, D; Ciaccio, R; Guccione, S
Combining molecular modelling with experimental methodologies: mechanism of membrane permeation and accumulation of ofloxacin
2002-01-01 Fresta, M; Guccione, S.; Beccari, A. R.; Furneri, P. M.; Puglisi, G.
Combining NMR and molecular modelling in a drug delivery context: investigation of the multi-mode inclusion of a new NPY-5 antagonist bromobenzenesulfonamide into beta-cyclodextrin
2004-01-01 Uccello-Barretta, G; Balzano, F; Sicoli, G; Friglola, C; Aldana, I; Monge, A; Paolino, D; Guccione, S
Design and synthesis of DNA-intercalating 9-fluoren-β-O-glycosides as potential IFN-inducers, and antiviral and cytostatic agents
2004-01-01 Arena, A; Neri, S; Ottanà, R; Ortuso, F; Pavone, B; Vigorita, M. G.; Alcaro, S
Design of 1-substituted 2-arylmethyl-4,5-methylenedioxybenzene derivatives as antiseizure agents
2004-01-01 Micale, N; De Sarro, G; Ferreri, G; Zappala, M; Grasso, S; Puia, G; De Micheli, C
Design, synthesis, and SAR analysis of novel selective sigma(1) ligands
2007-01-01 Collina, S; Loddo, G; Urbano, M; Linati, L; Callegari, A; Ortuso, F; Laggner, C; Langer, T; Prezzavento, O; Ronsisvalle, G; Azzolina, O; Alcaro, S
Design, synthesis, biophysical and biological studies of trisubstituted naphthalimides as G-quadruplex ligands
2011-01-01 Peduto, A; Pagano, B; Petronzi, C; Massa, A; Esposito, V; Virgilio, A; Paduano, F; Trapasso, F; Fiorito, F; Florio, S; Giancola, C; Galeone, A; Filosa, R
Development of 3-substituted-1H-indole derivatives as NR2B/NMDA receptor antagonists
2009-01-01 Gitto, R; Luca, Ld; Ferro, S; Citraro, R; Sarro, Gd; Costa, L; Ciranna, L; Chimirri, A
Evaluation of chromane derivatives: Promising privileged scaffolds for lead discovery within Alzheimer's disease
2022-01-01 Moutayakine, A.; Marques, C.; Lopez, O.; Bagetta, D.; Leitzbach, L.; Hagenow, S.; Carreiro, E. P.; Stark, H.; Alcaro, S.; Fernandez-Bolanos, J. G.; Burke, A. J.
Exploring new chemical functionalities to improve aromatase inhibition of steroids
2016-01-01 Varela, Cl; Amaral, C; Correia-da-Silva, G; Costa, Sc; Carvalho, Ra; Costa, G; Alcaro, S; Teixeira, Naa; Tavares-da-Silva, Ej; Roleira, Fmf
Identification of the stereochemical requirements in the 4-aryl-2-cycloalkylidenhydrazinylthiazole scaffold for the design of selective human monoamine oxidase B inhibitors.
2014-01-01 D'Ascenzio, M; Carradori, S; Secci, D; Mannina, L; Sobolev, Ap; De Monte, C; Cirilli, R; Yáñez, M; Ortuso, F; Alcaro, S
Investigations on the 2-thiazolylhydrazyne scaffold: synthesis and molecular modeling of selective human monoamine oxidase inhibitors
2010-01-01 Chimenti, F; Bolasco, A; Secci, D; Chimenti, P; Granese, A; Carradori, S; Yáñez, M; Orallo, F; Alcaro, S; Ortuso, F
Macrocyclic naphthalene diimides as G-quadruplex binders.
2015-01-01 Marchetti, C; Minarini, A; Tumiatti, V; Moraca, F; Parrotta, L; Alcaro, S; Rigo, R; Sissi, C; Gunaratnam, M; Ohnmacht, Sa; Neidle, S; Milelli, A.
N-Alkyl dien- and trienamides from the roots of Otanthus maritimus with binding affinity for opioid and cannabinoid receptors.
2013-01-01 Ruiu, S; Anzani, N; Orrù, A; Floris, C; Caboni, P; Maccioni, E; Distinto, S; Alcaro, S; Cottiglia, F.
Structure-activity relationships of 2-aryl-2,5-dihydropyridazino[4,3-b]indol-3(3H)-ones at the benzodiazepine receptor
1996-01-01 Palluotto, F; Carotti, A; Casini, G; Campagna, F; Genchi, G; Rizzo, M; De Sarro, G
Structure-guided design of new indoles as negative allosteric modulators (NAMs) of N-methyl-D-aspartate receptor (NMDAR) containing GluN2B subunit
2016-01-01 Buemi, Mr; De Luca, L; Ferro, S; Russo, E; Gitto, R; De Sarro, G
Synthesis and anticonvulsant evaluation of N-substituted isoquinoline AMPA receptor antagonists
2008-01-01 Gitto, R; DE LUCA, L; Pagano, B; Citraro, R; DE SARRO, G; Costa, L; Ciranna, L; Chimirri, A
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 2-Aryl-2,5-dihydropyridazino[4,3-b]indol-3(3H)-ones: novel rigid planar benzodiazepine receptor ligands. | 1-gen-1993 | Campagna, F; Carotti, A; Casini, G; Palluotto, F; Genchi, G; De Sarro, G | |
| A new series of flavones, thioflavones, and flavanones as selective monoamine oxidase-B inhibitors | 1-gen-2010 | Chimenti, F; Fioravanti, R; Bolasco, A; Chimenti, P; Secci, D; Rossi, F; Yáñez, M; Orallo, F; Alcaro, S; Cirilli, R; Ferretti, R; Sanna, M. L.; Ortuso, F | |
| Biocatalysed synthesis of β-O-glucosides from 9-fluorenon-2-carbohydroxyesters. Part 3: IFN-inducing and anti-HSV-2 properties | 1-gen-2005 | Arena, A; DI BELLA, R; Neri, S; Ottanà, R; Ortuso, F; Pavone, B; Trincone, A; Vigorita, M. G.; Alcaro, S | |
| Combined NMR-crystallographic and modelling investigation of the inclusion of molsidomine into alpha-, beta- and gamma-cyclodextrins | 1-gen-2005 | Uccello-Barretta, G; Balzano, F; Paolino, D; Ciaccio, R; Guccione, S | |
| Combining molecular modelling with experimental methodologies: mechanism of membrane permeation and accumulation of ofloxacin | 1-gen-2002 | Fresta, M; Guccione, S.; Beccari, A. R.; Furneri, P. M.; Puglisi, G. | |
| Combining NMR and molecular modelling in a drug delivery context: investigation of the multi-mode inclusion of a new NPY-5 antagonist bromobenzenesulfonamide into beta-cyclodextrin | 1-gen-2004 | Uccello-Barretta, G; Balzano, F; Sicoli, G; Friglola, C; Aldana, I; Monge, A; Paolino, D; Guccione, S | |
| Design and synthesis of DNA-intercalating 9-fluoren-β-O-glycosides as potential IFN-inducers, and antiviral and cytostatic agents | 1-gen-2004 | Arena, A; Neri, S; Ottanà, R; Ortuso, F; Pavone, B; Vigorita, M. G.; Alcaro, S | |
| Design of 1-substituted 2-arylmethyl-4,5-methylenedioxybenzene derivatives as antiseizure agents | 1-gen-2004 | Micale, N; De Sarro, G; Ferreri, G; Zappala, M; Grasso, S; Puia, G; De Micheli, C | |
| Design, synthesis, and SAR analysis of novel selective sigma(1) ligands | 1-gen-2007 | Collina, S; Loddo, G; Urbano, M; Linati, L; Callegari, A; Ortuso, F; Laggner, C; Langer, T; Prezzavento, O; Ronsisvalle, G; Azzolina, O; Alcaro, S | |
| Design, synthesis, biophysical and biological studies of trisubstituted naphthalimides as G-quadruplex ligands | 1-gen-2011 | Peduto, A; Pagano, B; Petronzi, C; Massa, A; Esposito, V; Virgilio, A; Paduano, F; Trapasso, F; Fiorito, F; Florio, S; Giancola, C; Galeone, A; Filosa, R | |
| Development of 3-substituted-1H-indole derivatives as NR2B/NMDA receptor antagonists | 1-gen-2009 | Gitto, R; Luca, Ld; Ferro, S; Citraro, R; Sarro, Gd; Costa, L; Ciranna, L; Chimirri, A | |
| Evaluation of chromane derivatives: Promising privileged scaffolds for lead discovery within Alzheimer's disease | 1-gen-2022 | Moutayakine, A.; Marques, C.; Lopez, O.; Bagetta, D.; Leitzbach, L.; Hagenow, S.; Carreiro, E. P.; Stark, H.; Alcaro, S.; Fernandez-Bolanos, J. G.; Burke, A. J. | |
| Exploring new chemical functionalities to improve aromatase inhibition of steroids | 1-gen-2016 | Varela, Cl; Amaral, C; Correia-da-Silva, G; Costa, Sc; Carvalho, Ra; Costa, G; Alcaro, S; Teixeira, Naa; Tavares-da-Silva, Ej; Roleira, Fmf | |
| Identification of the stereochemical requirements in the 4-aryl-2-cycloalkylidenhydrazinylthiazole scaffold for the design of selective human monoamine oxidase B inhibitors. | 1-gen-2014 | D'Ascenzio, M; Carradori, S; Secci, D; Mannina, L; Sobolev, Ap; De Monte, C; Cirilli, R; Yáñez, M; Ortuso, F; Alcaro, S | |
| Investigations on the 2-thiazolylhydrazyne scaffold: synthesis and molecular modeling of selective human monoamine oxidase inhibitors | 1-gen-2010 | Chimenti, F; Bolasco, A; Secci, D; Chimenti, P; Granese, A; Carradori, S; Yáñez, M; Orallo, F; Alcaro, S; Ortuso, F | |
| Macrocyclic naphthalene diimides as G-quadruplex binders. | 1-gen-2015 | Marchetti, C; Minarini, A; Tumiatti, V; Moraca, F; Parrotta, L; Alcaro, S; Rigo, R; Sissi, C; Gunaratnam, M; Ohnmacht, Sa; Neidle, S; Milelli, A. | |
| N-Alkyl dien- and trienamides from the roots of Otanthus maritimus with binding affinity for opioid and cannabinoid receptors. | 1-gen-2013 | Ruiu, S; Anzani, N; Orrù, A; Floris, C; Caboni, P; Maccioni, E; Distinto, S; Alcaro, S; Cottiglia, F. | |
| Structure-activity relationships of 2-aryl-2,5-dihydropyridazino[4,3-b]indol-3(3H)-ones at the benzodiazepine receptor | 1-gen-1996 | Palluotto, F; Carotti, A; Casini, G; Campagna, F; Genchi, G; Rizzo, M; De Sarro, G | |
| Structure-guided design of new indoles as negative allosteric modulators (NAMs) of N-methyl-D-aspartate receptor (NMDAR) containing GluN2B subunit | 1-gen-2016 | Buemi, Mr; De Luca, L; Ferro, S; Russo, E; Gitto, R; De Sarro, G | |
| Synthesis and anticonvulsant evaluation of N-substituted isoquinoline AMPA receptor antagonists | 1-gen-2008 | Gitto, R; DE LUCA, L; Pagano, B; Citraro, R; DE SARRO, G; Costa, L; Ciranna, L; Chimirri, A |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile